SCHEMBL8980460

SCHEMBL8980460

O=[C]CNC(=O)[C@@H](S)C(=O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.46
CES1 P23141 2/20 0.42
CES2 O00748 1/20 0.42
LMNA P02545 1/20 0.42
ALKBH5 Q6P6C2 1/20 0.40
PGR P06401 1/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
HTR2A P28223 1/20 0.40
HRH1 P35367 1/20 0.40
KCNH2 Q12809 1/20 0.40
MDM2 Q00987 1/20 0.40
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
ATM Q13315 3/20 0.39
GAA P10253 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HSP90AA1 P07900 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8595093 0.81 ACE (0.51) KMT2ALMNAALKBH5MDM2TDP1
SCHEMBL2028236 0.76 ACE (0.47) KMT2ALMNATDP1MAPTMAPK1
SCHEMBL7745199 0.76 ACE (0.47) KMT2ALMNATDP1MAPTMAPK1
SCHEMBL2417683 0.75 TDP1 (0.56) KMT2ACES1CES2LMNAALKBH5
SCHEMBL9067249 0.75 GPR139 (0.47) KMT2AMEN1ACE
SCHEMBL237683 0.74 GAA (0.63) LMNANPC1RAB9AGAASMN1; SMN2
SCHEMBL10720961 0.73 KMT2A (0.38) KMT2AMDM2NPC1RAB9AATM
SCHEMBL9067258 0.72 SLC1A1 (0.39) KMT2AACE
SCHEMBL5274104 0.72 TDP1 (0.52) CES1CES2LMNAALKBH5PGR
SCHEMBL7207824 0.72 TDP1 (0.52) CES1CES2LMNAALKBH5PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0710228-A1 HYDRAZINO-TYPE RADIONUCLIDE CHELATORS HAVING AN N 3?S CONFIGURATION RESOLUTION PHARMACEUTICALS INC. (CA) 1996-05-08 EP disclosed
WO-1995003280-A1 HYDRAZINO-TYPE RADIONUCLIDE CHELATORS HAVING AN N3S CONFIGURATION RESOLUTION PHARMACEUTICALS INC. (CA) 1995-02-02 WO disclosed