SCHEMBL8980925

SCHEMBL8980925

CCOC(=O)c1cccc(C(=O)CC)c1OCc1ccc(C(=O)c2ccccc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.60
HTT P42858 5/20 0.60
NPSR1 Q6W5P4 3/20 0.60
HPGD P15428 2/20 0.60
SMN1; SMN2 Q16637 4/20 0.57
MAPT P10636 2/20 0.57
GAA P10253 1/20 0.57
RAB9A P51151 1/20 0.57
CYP2C9 P11712 2/20 0.53
CYP2C19 P33261 2/20 0.53
L3MBTL1 Q9Y468 2/20 0.47
ATM Q13315 1/20 0.47
TSHR P16473 2/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
TP53 P04637 1/20 0.43
POLB P06746 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
PPARG P37231 1/20 0.43
MAPK10 P53779 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8980579 0.90 TSHR (0.53) ALDH1A1HTTNPSR1HPGDSMN1; SMN2
SCHEMBL8980703 0.88 ALDH1A1 (0.62) ALDH1A1HTTNPSR1HPGDSMN1; SMN2
SCHEMBL8980608 0.81 L3MBTL1 (0.55) HTTSMN1; SMN2MAPTGAARAB9A
SCHEMBL28877532 0.80 ALDH1A1 (0.56) ALDH1A1HTTHPGDL3MBTL1TSHR
SCHEMBL8980558 0.77 PTGER1 (0.50) ALDH1A1HTTHPGDSMN1; SMN2MAPT
SCHEMBL27968967 0.75 TSHR (0.53) ALDH1A1HTTHPGDL3MBTL1TSHR
SCHEMBL15716659 0.74 ALDH1A1 (0.67) ALDH1A1HTTNPSR1HPGDRAB9A
SCHEMBL28957917 0.73 TSHR (0.50) ALDH1A1RAB9AL3MBTL1TSHRCYP3A4
SCHEMBL8876258 0.73 TSHR (0.47) ALDH1A1HPGDSMN1; SMN2MAPTRAB9A
SCHEMBL1561432 0.72 PPIA (0.53) HTTNPSR1SMN1; SMN2MAPTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1132508-A Piperazine derivatives REORDATI IND CHIMICA E FARMACE (CH) 1996-10-02 CN disclosed
EP-0711288-A1 PIPERAZINE DERIVATIVES AS ALPHA 1A-ADRENERGIC RECEPTOR ANTAGONISTS RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA S.p.a. (IT) 1996-05-15 EP disclosed
WO-1995004049-A1 PIPERAZINE DERIVATIVES AS α1A-ADRENERGIC RECEPTOR ANTAGONISTS RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1995-02-09 WO disclosed