SCHEMBL8990012

SCHEMBL8990012

C[C@@H](C(=O)O)N(C)C(=O)CBr

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.33
LTA4H P09960 1/20 0.33
ALDH1A1 P00352 2/20 0.32
TRPA1 O75762 2/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11163798 0.81 FFAR3 (0.36) LTA4HALDH1A1TP53
SCHEMBL14753764 0.81 FFAR3 (0.36) LTA4HALDH1A1TP53
SCHEMBL1563864 0.78
SCHEMBL31589933 0.78 CHRNB2 (0.35) ALDH1A1
SCHEMBL11166642 0.77 LTA4H (0.40) LTA4HALDH1A1TP53
SCHEMBL9303262 0.77 ALDH1A1 (0.40) TSHRLTA4HALDH1A1TP53
SCHEMBL9302554 0.77 ALDH1A1 (0.40) TSHRLTA4HALDH1A1TP53
SCHEMBL17814865 0.77 LTA4H (0.36) LTA4HTP53
SCHEMBL31589523 0.77 KDM4C (0.36) ALDH1A1
SCHEMBL16006838 0.74 FOLH1 (0.32) LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5578633-A VASOPRESSIN AND OXYTOCIN ANTAGONISTS SANOFI (FR) 1996-11-26 US disclosed
US-5481005-A N-sulfonylindoline derivatives, their preparation and the pharmaceutical compositions in which they are present SANOFI (FR) 1996-01-02 US disclosed
US-5397801-A Affinity for vasopressin and ocytocin receptors; disorders of nervous, cardiovascular and gastrointestinal systems SANOFI (FR) 1995-03-14 US disclosed
US-5338755-A Have affinity for vasopressin and ocytocin receptors; intermediates for drugs that act on central nervous system ELF SANOFI (FR) 1994-08-16 US disclosed