SCHEMBL8990761

SCHEMBL8990761

Cc1ccc(CCNc2nc(N)c(N)c(N)n2)cc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.51
GALR3 O60755 1/20 0.51
ADORA2A P29274 5/20 0.50
ADORA1 P30542 4/20 0.50
ADORA2B P29275 3/20 0.50
ADORA3 P0DMS8 3/20 0.50
CA1 P00915 7/20 0.47
CA2 P00918 7/20 0.47
CA9 Q16790 7/20 0.47
TMIGD3 P0DMS9 1/20 0.44
MAPT P10636 1/20 0.44
ROCK1 Q13464 1/20 0.44
ADRA1D P25100 1/20 0.43
HTR2C P28335 1/20 0.43
HTR7 P34969 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
HTR6 P50406 1/20 0.43
TLR7 Q9NYK1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8990589 0.83 APP (0.71) APPADORA2AADORA1ADORA2BADORA3
SCHEMBL8990551 0.83 ADORA3 (0.61) APPADORA2AADORA1ADORA2BADORA3
Hydrochloric Acid SCHEMBL5471522 0.81 APP (0.69) APPADORA2AADORA1ADORA2BADORA3
SCHEMBL8990782 0.76 LMNA (0.71) APPADORA2AADORA1ADORA2BADORA3
Sulfuric Acid SCHEMBL5463730 0.75 APP (0.61) APPADORA2AADORA1ADORA2BADORA3
SCHEMBL5161863 0.74 ADORA2A (0.68) ADORA2AADORA1ADORA2BADORA3TMIGD3
SCHEMBL4373125 0.70 HTR7 (0.74) CA1CA2CA9ADRA1DHTR2C
SCHEMBL24756902 0.70 MAPT (0.65) APPGALR3CA1CA2CA9
SCHEMBL26267841 0.70 MAPT (0.65) APPGALR3CA1CA2CA9
SCHEMBL8547756 0.70 APP (0.76) APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5500428-A Furyl-substituted purines and adenosine antagonists IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1996-03-19 US disclosed
US-5300509-A Adenosine antagonists for treating cardiovascular disorders, vasodilation IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-04-05 US disclosed
EP-0544445-A2 Furyl-substituted purines, oxazolopyrimidines and pteridines as adenosine antagonists ZENECA LIMITED (GB) 1993-06-02 EP disclosed