SCHEMBL8990782

SCHEMBL8990782

COc1ccc(CCNc2nc(N)c(N)c(N)n2)cc1OC

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.71
TSHR P16473 2/20 0.71
ADORA2A P29274 2/20 0.60
POLB P06746 3/20 0.59
ALOX15 P16050 2/20 0.59
USP2 O75604 1/20 0.59
CRHBP P24387 1/20 0.59
CRHR2 Q13324 1/20 0.59
NPSR1 Q6W5P4 1/20 0.59
ADORA3 P0DMS8 1/20 0.58
ADORA2B P29275 1/20 0.58
ADORA1 P30542 1/20 0.58
MAPT P10636 4/20 0.57
TP53 P04637 3/20 0.57
KMT2A Q03164 2/20 0.57
MEN1 O00255 1/20 0.57
GAA P10253 3/20 0.56
ATM Q13315 1/20 0.55
APP P05067 3/20 0.55
BCHE P06276 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9008391 0.88 LMNA (0.83) LMNATSHRPOLBALOX15USP2
SCHEMBL9008401 0.82 LMNA (0.72) LMNATSHRPOLBALOX15USP2
SCHEMBL14028292 0.82 TSHR (0.72) LMNATSHRPOLBALOX15USP2
SCHEMBL8990551 0.81 ADORA3 (0.61) LMNATSHRADORA2AADORA3ADORA2B
SCHEMBL5161859 0.78 ADORA2A (0.58) LMNATSHRADORA2APOLBALOX15
SCHEMBL9008399 0.77 SMN1; SMN2 (0.67) LMNATSHRPOLBALOX15USP2
SCHEMBL8990761 0.76 APP (0.51) ADORA2AADORA3ADORA2BADORA1MAPT
SCHEMBL1581342 0.74 ATM (0.67) LMNATSHRPOLBMAPTKMT2A
SCHEMBL1513260 0.74 APP (0.60) LMNATSHRPOLBMAPTTP53
SCHEMBL7435099 0.73 ATM (0.76) POLBALOX15MAPTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5500428-A Furyl-substituted purines and adenosine antagonists IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1996-03-19 US disclosed
US-5300509-A Adenosine antagonists for treating cardiovascular disorders, vasodilation IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-04-05 US disclosed
EP-0544445-A2 Furyl-substituted purines, oxazolopyrimidines and pteridines as adenosine antagonists ZENECA LIMITED (GB) 1993-06-02 EP disclosed