SCHEMBL8990955

SCHEMBL8990955

CCOc1nc(-c2ccco2)oc1C(C)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.43
NPC1 O15118 5/20 0.43
RECQL P46063 1/20 0.43
HSD17B10 Q99714 9/20 0.43
ALDH1A1 P00352 9/20 0.43
KDM4E B2RXH2 8/20 0.43
HPGD P15428 8/20 0.43
MAPT P10636 6/20 0.43
TSHR P16473 5/20 0.43
TP53 P04637 4/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
GAA P10253 3/20 0.43
LMNA P02545 3/20 0.40
MAPK1 P28482 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
ALOX15 P16050 2/20 0.40
HTT P42858 1/20 0.40
POLB P06746 2/20 0.39
PPARG P37231 2/20 0.39
PPARA Q07869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8990667 0.83 HPGD (0.44) RAB9ANPC1RECQLHSD17B10ALDH1A1
SCHEMBL8990962 0.76 RAB9A (0.43) RAB9ANPC1RECQLHSD17B10ALDH1A1
SCHEMBL8990670 0.70 ALDH1A1 (0.43) RAB9ANPC1RECQLHSD17B10ALDH1A1
SCHEMBL27558918 0.67 ALDH1A1 (0.48) RAB9ANPC1HSD17B10ALDH1A1KDM4E
SCHEMBL8990569 0.67 RAB9A (0.48) RAB9ANPC1RECQLHSD17B10ALDH1A1
SCHEMBL28295524 0.66 TARBP2 (0.62) HSD17B10ALDH1A1KDM4EHPGDTSHR
SCHEMBL27545042 0.62 RAB9A (0.51) RAB9ANPC1RECQLHSD17B10ALDH1A1
SCHEMBL12611216 0.62 SLC1A3 (0.61) HSD17B10ALDH1A1HPGDMAPTTSHR
SCHEMBL10504755 0.62 KDM4E (0.51) RAB9ANPC1HSD17B10ALDH1A1KDM4E
SCHEMBL3436254 0.62 L3MBTL1 (0.58) RAB9ANPC1HSD17B10ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5500428-A Furyl-substituted purines and adenosine antagonists IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1996-03-19 US disclosed
US-5300509-A Adenosine antagonists for treating cardiovascular disorders, vasodilation IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-04-05 US disclosed
EP-0544445-A2 Furyl-substituted purines, oxazolopyrimidines and pteridines as adenosine antagonists ZENECA LIMITED (GB) 1993-06-02 EP disclosed