SCHEMBL8991022

SCHEMBL8991022

COc1ccc(Cn2c(N)c(SC(N)=O)c3c(N)ncnc32)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.44
HSD17B10 Q99714 4/20 0.44
ALDH1A1 P00352 3/20 0.44
GLA P06280 3/20 0.44
GAA P10253 3/20 0.44
HPGD P15428 3/20 0.44
CASP1 P29466 3/20 0.44
CASP7 P55210 3/20 0.44
MAPK1 P28482 2/20 0.42
USP2 O75604 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
EGFR P00533 3/20 0.41
RET P07949 1/20 0.40
PDE8B O95263 1/20 0.40
PDE1B Q01064 5/20 0.39
ABL1 P00519 3/20 0.39
SRC P12931 3/20 0.39
PIK3CD O00329 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8991328 0.89 ALDH1A1 (0.44) KDM4EHSD17B10ALDH1A1GLAGAA
SCHEMBL8991429 0.85 MAPK1 (0.54) KDM4EHSD17B10ALDH1A1GAAHPGD
SCHEMBL8991185 0.85 KDM4E (0.41) KDM4EHSD17B10MAPK1TSHRHTT
SCHEMBL8991284 0.81 KDM4E (0.44) KDM4EHSD17B10ALDH1A1GLAGAA
SCHEMBL8991108 0.81 KDM4E (0.46) KDM4EHSD17B10ALDH1A1HPGDMAPK1
SCHEMBL8991011 0.80 KDM4E (0.49) KDM4EHSD17B10ALDH1A1GLAGAA
SCHEMBL8991267 0.79 KDM4E (0.48) KDM4EHSD17B10ALDH1A1GLAGAA
SCHEMBL7705468 0.79 EGFR (0.43) EGFRPDE8BABL1SRCKDR
SCHEMBL8991491 0.77 HTT (0.42) KDM4EHSD17B10ALDH1A1MAPK1NPSR1
SCHEMBL8991147 0.77 GAA (0.39) KDM4EHSD17B10ALDH1A1GAAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5543413-A VIRAL ACTIVITY AGAINST HUMAN CYTOMEGALOVIRUS AND HERPES SIMPLEX VIRUS REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 1996-08-06 US disclosed