SCHEMBL8991244

SCHEMBL8991244

CNc1ncnc2c1c(SC(N)=O)cn2Cc1ccc(C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
GAA P10253 1/20 0.39
TP53 P04637 4/20 0.37
MAPT P10636 4/20 0.37
SLC29A1 Q99808 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8991110 0.90 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL8991272 0.89 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DTP53
SCHEMBL8991207 0.88 AURKA (0.40) PDE4APDE4BPDE4CPDE4DTP53
SCHEMBL7698505 0.86 FYN (0.39) TP53MAPTSLC29A1ALDH1A1KDM4E
SCHEMBL8991419 0.83 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL8991078 0.81 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DGAA
SCHEMBL8991063 0.79 GAA (0.41) PDE4APDE4BPDE4CPDE4DGAA
SCHEMBL8991231 0.79 GAA (0.41) PDE4APDE4BPDE4CPDE4DGAA
SCHEMBL8991147 0.79 GAA (0.39) PDE4APDE4BPDE4CPDE4DGAA
SCHEMBL7700322 0.78 ADK (0.33) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5543413-A VIRAL ACTIVITY AGAINST HUMAN CYTOMEGALOVIRUS AND HERPES SIMPLEX VIRUS REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 1996-08-06 US disclosed