SCHEMBL8992651

SCHEMBL8992651

CC(C)(C)OC(=O)N(CCc1ccccc1)C(=O)Nc1cc(C(=O)OCc2ccccc2)cc(C(=O)OCc2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.47
KMT2A Q03164 2/20 0.42
GAA P10253 2/20 0.42
SLC6A2 P23975 1/20 0.41
SLC6A3 Q01959 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
HPGD P15428 1/20 0.40
KDM4E B2RXH2 1/20 0.40
NPY5R Q15761 1/20 0.39
LMNA P02545 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CASR P41180 2/20 0.38
BACE1 P56817 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
NCOR2 Q9Y618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8129548 0.98 RAB9A (0.45) RAB9AKMT2AGAASLC6A2SLC6A3
SCHEMBL8992582 0.92 RAB9A (0.58) RAB9AKMT2AGAASLC6A2SLC6A3
SCHEMBL8903055 0.91 RAB9A (0.42) RAB9AKMT2AGAASLC6A2SLC6A3
SCHEMBL8663889 0.89 ACE (0.49)
SCHEMBL8992625 0.84 ALDH1A1 (0.48) RAB9AKMT2AGAASLC6A2SLC6A3
SCHEMBL8992691 0.83 NPY5R (0.51) RAB9AKMT2AALDH1A1MAPTNPY5R
SCHEMBL8472195 0.82 NPY5R (0.59) RAB9AKMT2AGAASLC6A2SLC6A3
SCHEMBL8650559 0.80 RAB9A (0.56) RAB9AKMT2AGAASLC6A2SLC6A3
SCHEMBL30503476 0.74 CTSK (0.43) RAB9AGAAMAPTNPY5RL3MBTL1
Methylamine SCHEMBL8548886 0.73 L3MBTL1 (0.40) NPY5RL3MBTL1HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0719251-A1 BICYCLO (2.2.2) OCTANE DERIVATIVES CHOLECYSTOKININ AND/OR GASTRIN ANTAGONISTS JAMES BLACK FOUNDATION LIMITED (GB) 1996-07-03 EP disclosed
WO-1995005359-A1 BICYCLO (2.2.2) OCTANE DERIVATIVES CHOLECYSTOKININ AND/OR GASTRIN ANTAGONISTS JAMES BLACK FOUNDATION LIMITED (GB) 1995-02-23 WO disclosed