SCHEMBL8992798

SCHEMBL8992798

Cc1cccc(Cc2ccc(CC#N)cc2C)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.41
KDM4E B2RXH2 2/20 0.39
MMP3 P08254 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
IDO1 P14902 2/20 0.37
MPO P05164 1/20 0.36
DAO P14920 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
LTA4H P09960 1/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
FFAR1 O14842 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8093981 0.85 TAAR1 (0.46) TAAR1IDO1MPODAOLTA4H
SCHEMBL625612 0.83 ENPP2 (0.53) ENPP2KDM4EMMP3TAAR1IDO1
SCHEMBL8993099 0.83 CNR2 (0.44) ENPP2CNR1CNR2
SCHEMBL8992807 0.83 CNR2 (0.46) TAAR1IDO1CNR1CNR2
SCHEMBL8992963 0.82 LTA4H (0.46) ENPP2KDM4EMMP3TAAR1IDO1
SCHEMBL8085589 0.81 LTA4H (0.44) TAAR1IDO1LTA4H
SCHEMBL8992935 0.80 TAAR1 (0.41) TAAR1IDO1MPODAOLTA4H
SCHEMBL8993034 0.80 TAAR1 (0.41) TAAR1IDO1MPODAOCNR1
SCHEMBL2977626 0.77 ENPP2 (0.47) ENPP2KDM4EMMP3TAAR1IDO1
SCHEMBL18052640 0.75 ENPP2 (0.37) ENPP2KDM4EMMP3TDP1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed