SCHEMBL8992842

SCHEMBL8992842

O=C(O)C(C(=O)O)(C(=O)O)N1CCNCCNCCN(Cc2ccc(N=C=S)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 11/20 0.41
CHRM1 P11229 2/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
CHRM2 P08172 1/20 0.41
ADRA2C P18825 1/20 0.41
CCR2 P41597 1/20 0.41
CXCL12 P48061 1/20 0.41
BLM P54132 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
SLC2A1 P11166 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2B Q13224 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
OPRD1 P41143 1/20 0.36
KDM5C P41229 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18039301 0.83 CXCR4 (0.57) CXCR4CHRM1KMT2AMEN1CHRM2
SCHEMBL14312212 0.83 SIGMAR1 (0.46) CXCR4CHRM1KMT2AMEN1CHRM2
SCHEMBL8038136 0.82 SIGMAR1 (0.62) CXCR4CHRM1KMT2AMEN1CHRM2
SCHEMBL5745082 0.82 SIGMAR1 (0.54) CXCR4CHRM1KMT2AMEN1CHRM2
SCHEMBL8992770 0.82 CXCR4 (0.47) CXCR4CHRM1KMT2AMEN1CHRM2
SCHEMBL14312255 0.78 CXCR4 (0.50) CXCR4CHRM1KMT2AMEN1CHRM2
SCHEMBL10574436 0.78 ALDH1A1 (0.54) TDP1ALDH1A1LMNA
SCHEMBL8689068 0.78 CXCR4 (0.70) CXCR4CHRM1KMT2AMEN1CHRM2
SCHEMBL8038145 0.75 GRIN1 (0.48) CHRM1HRH3GRIN1GRIN2AGRIN2B
SCHEMBL16656265 0.75 GRIN1 (0.48) CHRM1HRH3GRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292689-B1 Substituted 1,4,7-triscarboxymethyl-1,4,7,10-tetraazacyclo-dodecane and analogs BRACCO INT BV (NL) 1996-07-31 EP claimed
US-4885363-A RADIOPHARMACEUTICAL IMAGING; MEDICAL DIAGNOSIS E. R. SQUIBB & SONS, INC. (US) 1989-12-05 US claimed
EP-0292689-A2 Substituted 1,4,7-triscarboxymethyl-1,4,7,10-tetraazacyclo-dodecane and analogs BRACCO INTERNATIONAL B.V. (NL) 1988-11-30 EP claimed