SCHEMBL8992770

SCHEMBL8992770

Nc1ccc(CN2CCNCCNCCN(C(C(=O)O)(C(=O)O)C(=O)O)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 11/20 0.47
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
ADRA2C P18825 1/20 0.47
CCR2 P41597 1/20 0.47
CXCL12 P48061 1/20 0.47
BLM P54132 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
SIGMAR1 Q99720 2/20 0.47
LMNA P02545 2/20 0.44
ALDH1A1 P00352 2/20 0.43
SLC2A1 P11166 1/20 0.39
PLK4 O00444 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8038136 0.88 SIGMAR1 (0.62) CXCR4KMT2AMEN1CHRM2CHRM1
SCHEMBL4019574 0.84 CXCR4 (0.52) CXCR4KMT2AMEN1CHRM2CHRM1
SCHEMBL10574436 0.83 ALDH1A1 (0.54) TDP1LMNAALDH1A1
SCHEMBL8992842 0.82 CXCR4 (0.41) CXCR4KMT2AMEN1CHRM2CHRM1
SCHEMBL8715048 0.81 CXCR4 (0.68) CXCR4KMT2AMEN1CHRM2CHRM1
SCHEMBL14478352 0.80 SIGMAR1 (0.53) CXCR4KMT2AMEN1CHRM2CHRM1
SCHEMBL1578113 0.79 SIGMAR1 (0.66) CXCR4KMT2AMEN1CHRM2CHRM1
SCHEMBL14478353 0.75 CXCR4 (0.57) CXCR4KMT2AMEN1CHRM2CHRM1
SCHEMBL8993114 0.74 KDM4E (0.39) SIGMAR1ALDH1A1
SCHEMBL28434277 0.74 SIGMAR1 (0.39) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292689-B1 Substituted 1,4,7-triscarboxymethyl-1,4,7,10-tetraazacyclo-dodecane and analogs BRACCO INT BV (NL) 1996-07-31 EP claimed
US-4885363-A RADIOPHARMACEUTICAL IMAGING; MEDICAL DIAGNOSIS E. R. SQUIBB & SONS, INC. (US) 1989-12-05 US claimed
EP-0292689-A2 Substituted 1,4,7-triscarboxymethyl-1,4,7,10-tetraazacyclo-dodecane and analogs BRACCO INTERNATIONAL B.V. (NL) 1988-11-30 EP claimed