SCHEMBL8992843

SCHEMBL8992843

COc1cc(OC)cc(C(O)c2ccc(C3OCCO3)cc2)c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.39
CREBBP Q92793 1/20 0.39
REN P00797 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
ALDH1A1 P00352 3/20 0.35
ALOX5 P09917 1/20 0.33
PTPN1 P18031 1/20 0.33
PPARG P37231 1/20 0.33
PPARD Q03181 1/20 0.33
FGFR1 P11362 2/20 0.33
FGFR2 P21802 2/20 0.33
FGFR4 P22455 2/20 0.33
FGFR3 P22607 2/20 0.33
CYP3A4 P08684 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3571617 0.81 ALDH1A1 (0.47) ALDH1A1PPARGPPARDSMN1; SMN2
SCHEMBL8021420 0.79 ALDH1A1 (0.38) BRD4CREBBPNPC1RAB9AALDH1A1
SCHEMBL2200862 0.75 ALDH1A1 (0.48) NPC1RAB9AALDH1A1FGFR1FGFR2
SCHEMBL4723773 0.75 MAOA (0.48) NPC1RAB9AMAPTKMT2ASMN1; SMN2
SCHEMBL1818480 0.75 ALDH1A1 (0.58) BRD4CREBBPALDH1A1CYP3A4KMT2A
SCHEMBL3569410 0.74 MAPK1 (0.47) BRD4ALDH1A1
SCHEMBL19903859 0.74 RAB9A (0.36) NPC1RAB9AALDH1A1ALOX5PTPN1
SCHEMBL3543214 0.74 ABL1 (0.55) BRD4CREBBPNPC1RAB9AALDH1A1
SCHEMBL9222651 0.73 NPC1 (0.30) NPC1RAB9ASMN1; SMN2
SCHEMBL5730369 0.73 TUBB4A (0.31) NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed