SCHEMBL8992912

SCHEMBL8992912

Cc1cccc(Cc2ccc(O)cc2C)c1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.48
ALOX5 P09917 2/20 0.47
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
IDO1 P14902 2/20 0.44
TAAR1 Q96RJ0 1/20 0.42
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
MAOB P27338 1/20 0.41
GPR84 Q9NQS5 1/20 0.40
IDH1 O75874 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5645276 0.86 ACHE (0.48) ACHEALOX5CYP1A2CYP2C19TAAR1
SCHEMBL27550232 0.84 ALOX5 (0.67) ALOX5
SCHEMBL8093981 0.84 TAAR1 (0.46) ACHEIDO1TAAR1CNR1CNR2
SCHEMBL8993034 0.81 TAAR1 (0.41) IDO1TAAR1CNR1CNR2
SCHEMBL7641239 0.80 MEN1 (0.49) ACHEALOX5CYP1A2CYP2C19
SCHEMBL29133193 0.80 ACHE (0.46) ACHEALOX5CYP1A2CYP2C19IDO1
SCHEMBL2094961 0.80 TAAR1 (0.48) ACHECYP2C19IDO1TAAR1
SCHEMBL11200939 0.80 ESR2 (0.52) ALOX5
SCHEMBL18174858 0.80 ACHE (0.64) ACHECYP1A2IDO1TAAR1GPR84
SCHEMBL8085589 0.79 LTA4H (0.44) CYP2C19IDO1TAAR1IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed