SCHEMBL8992923

SCHEMBL8992923

COc1cccc(Cc2ccc(C3OCCO3)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 3/20 0.48
MTNR1A P48039 1/20 0.45
MTNR1B P49286 1/20 0.45
CHRM2 P08172 1/20 0.44
CHRM1 P11229 1/20 0.44
CHRM3 P20309 1/20 0.44
HTR1B P28222 1/20 0.44
TAAR1 Q96RJ0 3/20 0.43
IDO1 P14902 2/20 0.43
AGXT P21549 2/20 0.43
ALDH1A1 P00352 1/20 0.43
SIGMAR1 Q99720 2/20 0.42
SLC5A1 P13866 1/20 0.42
SLC5A2 P31639 1/20 0.42
MAOB P27338 1/20 0.41
KDM1A O60341 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18063537 0.78 HTR2C (0.51) KDM1A
SCHEMBL16388357 0.78 CALM1 (0.48) LTA4HCHRM2CHRM3
SCHEMBL14191204 0.78 LTA4H (0.70) LTA4HMTNR1AMTNR1BCHRM2CHRM1
SCHEMBL8993057 0.78 LTA4H (0.43) LTA4HTAAR1IDO1AGXTSIGMAR1
SCHEMBL2099512 0.78 CHRM2 (0.66) LTA4HCHRM2CHRM1CHRM3HTR1B
SCHEMBL31739258 0.76 LTA4H (0.67) LTA4HMTNR1AMTNR1BCHRM2CHRM1
SCHEMBL2092574 0.76 LTA4H (0.67) LTA4HMTNR1AMTNR1BCHRM2CHRM1
SCHEMBL8093299 0.75 MTNR1A (0.57) LTA4HMTNR1AMTNR1BCHRM2CHRM1
SCHEMBL13880096 0.75 MAOB (0.62) LTA4HMTNR1AMTNR1BCHRM2CHRM1
SCHEMBL27950339 0.74 EED (0.50) CHRM2CHRM1CHRM3TAAR1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed