SCHEMBL8993038

SCHEMBL8993038

COc1cccc(Cc2ccc(CO)cc2)c1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.56
MTNR1B P49286 1/20 0.56
LTA4H P09960 3/20 0.53
CHRM2 P08172 1/20 0.53
CHRM1 P11229 1/20 0.53
CHRM3 P20309 1/20 0.53
TAAR1 Q96RJ0 3/20 0.51
IDO1 P14902 2/20 0.51
AGXT P21549 2/20 0.51
MAOB P27338 2/20 0.49
IDH1 O75874 1/20 0.48
HTR1B P28222 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14191204 0.87 LTA4H (0.70) MTNR1AMTNR1BLTA4HCHRM2CHRM1
SCHEMBL29587500 0.87 TAAR1 (0.60) CHRM2CHRM1CHRM3TAAR1IDO1
SCHEMBL96382 0.87 TAAR1 (0.60) CHRM2CHRM1CHRM3TAAR1IDO1
SCHEMBL2099512 0.87 CHRM2 (0.66) LTA4HCHRM2CHRM1CHRM3TAAR1
SCHEMBL31298122 0.86 LTA4H (0.63) MTNR1AMTNR1BLTA4HIDO1
SCHEMBL31739258 0.85 LTA4H (0.67) MTNR1AMTNR1BLTA4HCHRM2CHRM1
SCHEMBL2092574 0.85 LTA4H (0.67) MTNR1AMTNR1BLTA4HCHRM2CHRM1
SCHEMBL8093299 0.84 MTNR1A (0.57) MTNR1AMTNR1BLTA4HCHRM2CHRM1
SCHEMBL13880096 0.84 MAOB (0.62) MTNR1AMTNR1BLTA4HCHRM2CHRM1
SCHEMBL8993248 0.83 CALM1 (0.59) MTNR1AMTNR1BLTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed