SCHEMBL8993248

SCHEMBL8993248

COc1cc(Cc2ccc(CO)cc2)cc(OC)c1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CALM1 P0DP23 5/20 0.59
AKR1B1 P15121 1/20 0.49
LTA4H P09960 2/20 0.48
CYP19A1 P11511 1/20 0.47
ALDH1A1 P00352 1/20 0.44
SAE1 Q9UBE0 1/20 0.43
UBA2 Q9UBT2 1/20 0.43
CA2 P00918 1/20 0.41
ERN1 O75460 1/20 0.40
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11791322 0.86 CALM1 (0.55) CALM1AKR1B1CYP19A1ALDH1A1CA2
SCHEMBL8993364 0.85 LTA4H (0.65) CALM1LTA4HALDH1A1SAE1UBA2
SCHEMBL8993038 0.83 MTNR1A (0.56) LTA4HMTNR1AMTNR1B
SCHEMBL65276 0.83 ALDH1A1 (0.58) CALM1AKR1B1CYP19A1ALDH1A1
SCHEMBL5252553 0.82 ALDH1A1 (0.65) CALM1AKR1B1LTA4HCYP19A1ALDH1A1
SCHEMBL19352719 0.82 CALM1 (0.56) CALM1AKR1B1LTA4HCYP19A1ALDH1A1
SCHEMBL28123040 0.81 ALDH1A1 (0.55) CALM1AKR1B1CYP19A1ALDH1A1
SCHEMBL8993062 0.80 CALM1 (0.54) CALM1AKR1B1LTA4HCYP19A1ALDH1A1
SCHEMBL26784208 0.80 ABL1 (0.62) AKR1B1ERN1MTNR1AMTNR1B
SCHEMBL11810459 0.79 LTA4H (0.69) CALM1LTA4HCYP19A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed