SCHEMBL8993074

SCHEMBL8993074

COc1cccc(Cc2ccc(-c3c[nH]nc3N)cc2OC)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.49
FGFR1 P11362 1/20 0.44
FGFR4 P22455 1/20 0.44
LTA4H P09960 1/20 0.44
FYN P06241 2/20 0.42
GPR55 Q9Y2T6 2/20 0.41
CNR1 P21554 1/20 0.41
PRKCI P41743 1/20 0.41
PRKCZ Q05513 1/20 0.41
KCNH2 Q12809 1/20 0.41
HTR1B P28222 1/20 0.40
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
CNR2 P34972 2/20 0.39
ADCY10 Q96PN6 1/20 0.39
PDCD1 Q15116 1/20 0.39
CD274 Q9NZQ7 1/20 0.39
IDO1 P14902 1/20 0.39
AGXT P21549 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8992949 0.88 DHFR (0.49) DHFRFGFR1FGFR4LTA4HGPR55
SCHEMBL8992951 0.84 LTA4H (0.57) DHFRFGFR1FGFR4LTA4HHTR1B
SCHEMBL4700185 0.78 TDO2 (0.55) FYN
SCHEMBL25798793 0.71 ABCB1 (0.62) DHFRGPR55CNR1CNR2
SCHEMBL8993377 0.71 CNR1 (0.49) DHFRGPR55CNR1CNR2IDO1
SCHEMBL27289914 0.70 FGFR1 (0.49) DHFRFGFR1FGFR4HTR1B
SCHEMBL8992845 0.70 FYN (0.40) DHFRFGFR1FGFR4FYNGPR55
SCHEMBL8992903 0.70 FYN (0.40) DHFRFGFR1FGFR4FYNGPR55
SCHEMBL8992834 0.69 LTA4H (0.53) LTA4HROCK2ROCK1IDO1TAAR1
SCHEMBL28438782 0.68 DHFR (0.63) DHFRFGFR1FGFR4LTA4HHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed