SCHEMBL8992834

SCHEMBL8992834

Cc1cccc(Cc2ccc(-c3c[nH]nc3N)cc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.53
MPO P05164 2/20 0.42
IDO1 P14902 2/20 0.41
ROCK2 O75116 2/20 0.39
PLK4 O00444 1/20 0.39
AURKA O14965 1/20 0.39
JAK2 O60674 1/20 0.39
CHEK2 O96017 1/20 0.39
NTRK1 P04629 1/20 0.39
CDK1 P06493 1/20 0.39
CSF1R P07333 1/20 0.39
PRKACA P17612 1/20 0.39
FLT1 P17948 1/20 0.39
RPS6KB1 P23443 1/20 0.39
CDK2 P24941 1/20 0.39
MARK3 P27448 1/20 0.39
AKT1 P31749 1/20 0.39
FLT4 P35916 1/20 0.39
KDR P35968 1/20 0.39
FLT3 P36888 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8993365 0.84 MPO (0.44) LTA4HMPOIDO1ROCK2TAAR1
SCHEMBL8992951 0.84 LTA4H (0.57) LTA4HIDO1BRS3TAAR1
SCHEMBL8993116 0.84 LTA4H (0.45) LTA4HMPOROCK2JAK2CSF1R
SCHEMBL11743569 0.79 LRRK2 (0.49) IDO1NTRK1CSF1RPRKACAKDR
SCHEMBL8093804 0.74 TAAR1 (0.56) LTA4HIDO1TAAR1DAO
SCHEMBL20067936 0.73 TAAR1 (0.57) LTA4HMPOIDO1TAAR1DAO
SCHEMBL8992896 0.73 MPO (0.47) MPOCHEK2TAAR1ALDH1A1CYP3A4
SCHEMBL27681631 0.72 LTA4H (0.55) LTA4HIDO1TAAR1CA1CA2
SCHEMBL8992949 0.71 DHFR (0.49) LTA4HIDO1TAAR1
SCHEMBL8085716 0.71 CALM1 (0.55) LTA4HIDO1TAAR1DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1036919-C Pyrazole condensed ring derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMA CO LTD (JP) 1998-01-07 CN disclosed
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed