SCHEMBL8993250

SCHEMBL8993250

Cc1ccc(Cc2ccc(CC#N)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.41
CYP2A6 P11509 2/20 0.41
ALDH1A1 P00352 2/20 0.41
IDO1 P14902 1/20 0.41
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
MAPT P10636 2/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
CYP1A2 P05177 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
KMT2A Q03164 1/20 0.37
LTA4H P09960 1/20 0.37
AGXT P21549 2/20 0.37
TDP1 Q9NUW8 2/20 0.36
ACHE P22303 1/20 0.36
GLA P06280 1/20 0.36
NPC1 O15118 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL247479 0.93 CYP2A6 (0.46) CYP2A6ALDH1A1IDO1L3MBTL1MAPT
SCHEMBL8763328 0.88 KMT2A (0.42) ALDH1A1L3MBTL1MAPTCYP1A2KMT2A
SCHEMBL9925859 0.86 NAAA (0.44) CYP2A6ALDH1A1IDO1L3MBTL1MAPT
Toluene SCHEMBL15756051 0.84 LMNA (0.48) CYP2A6ALDH1A1IDO1L3MBTL1MAPT
Toluene SCHEMBL15303842 0.84 LMNA (0.48) CYP2A6ALDH1A1IDO1L3MBTL1MAPT
Toluene SCHEMBL15756043 0.84 LMNA (0.48) CYP2A6ALDH1A1IDO1L3MBTL1MAPT
SCHEMBL4193868 0.81 MMP3 (0.43) CYP2A6ALDH1A1IDO1L3MBTL1MAPT
SCHEMBL8992963 0.81 LTA4H (0.46) IDO1POLBTAAR1KMT2ALTA4H
SCHEMBL1149394 0.80 IDO1 (0.58) SRD5A2CYP2A6ALDH1A1IDO1CYP1A2
SCHEMBL2154504 0.80 KMT2A (0.47) CYP2A6L3MBTL1MAPTGAACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed