SCHEMBL8993484

SCHEMBL8993484

CCSc1ccc(C(=O)O)c(Cl)c1OCCOC

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKAB2 O43741 1/20 0.36
PRKAG1 P54619 1/20 0.36
PRKAA2 P54646 1/20 0.36
PRKAA1 Q13131 1/20 0.36
PRKAG3 Q9UGI9 1/20 0.36
PRKAG2 Q9UGJ0 1/20 0.36
PRKAB1 Q9Y478 1/20 0.36
ALDH1A1 P00352 4/20 0.34
PKM P14618 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PTGER4 P35408 1/20 0.34
HPGD P15428 4/20 0.33
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 2/20 0.32
MAPT P10636 2/20 0.32
APEX1 P27695 1/20 0.32
ABL1 P00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8993574 0.80 ALDH1A1 (0.44) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL24886357 0.80 HPGD (0.45) ALDH1A1TDP1HPGDKMT2ASMN1; SMN2
SCHEMBL6562605 0.77 THRB (0.44) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL8993535 0.76 MAPT (0.45) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL7976218 0.75 PRKAB2 (0.37) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL9751862 0.74 MAPK1 (0.36) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL9709807 0.74 ALDH1A1 (0.39) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL24886348 0.71 HPGD (0.41) ALDH1A1HPGDMEN1KMT2ASMN1; SMN2
SCHEMBL8993452 0.71 NPC1 (0.33) ALDH1A1TDP1ABL1TSHRRECQL
SCHEMBL8493043 0.71 TDP1 (0.41) ALDH1A1PKMTDP1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0369803-B2 Trisubstituted benzoic acid intermediates ZENECA INC (US) 1996-08-14 EP disclosed
EP-0444152-B1 CERTAIN 2-(2',3',4'-TRISUBSTITUTED BENZOYL)-1,3-CYCLOHEXANEDIONES ZENECA INC (US) 1995-06-14 EP disclosed
EP-0444143-B1 TRISUBSTITUTED BENZOIC ACID INTERMEDIATES ZENECA INC (US) 1994-11-30 EP disclosed
US-5075497-A Chemical intermediate for 2-(2,3,4-trisubstitutedbenzoyl)-1,3-cyclohexanedione ICI AMERICAS, INC. (US) 1991-12-24 US disclosed
US-5073642-A Trisubstituted benzoic acid intermediates ICI AMERICAS INC. (US) 1991-12-17 US disclosed
US-5068423-A Intermediates for herbicides 2-(2,3,4-trisubstituted benzoyl)-1,3-cyclohexanediones ICI AMERICAS INC. (US) 1991-11-26 US disclosed
US-5047572-A For 2-*2,3,4-trisubstituted benzoyl)-1,3-cyclohexanedione ICI AMERICAS INC. (US) 1991-09-10 US disclosed
US-5001256-A Trisubstituted benzoic acid intermediates ICI AMERICAS INC. (US) 1991-03-19 US disclosed
US-4957538-A HERBICIDES ICI AMERICAS INC. (US) 1990-09-18 US disclosed
WO-1990005715-A1 TRISUBSTITUTED BENZOIC ACID INTERMEDIATES ICI AMERICAS INC. (US) 1990-05-31 WO disclosed
WO-1990005712-A1 CERTAIN 2-(2',3',4'-TRISUBSTITUTED BENZOYL)-1,3-CYCLOHEXANEDIONES ICI AMERICAS INC. (US) 1990-05-31 WO disclosed
EP-0369803-A1 Trisubstituted benzoic acid intermediates ZENECA INC. (US) 1990-05-23 EP disclosed