SCHEMBL8995206

SCHEMBL8995206

CN(C)COc1ccc([C]=O)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.40
ESR2 Q92731 2/20 0.40
CXCR1 P25024 4/20 0.39
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
HRH3 Q9Y5N1 3/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
NQO1 P15559 1/20 0.36
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
LTA4H P09960 1/20 0.35
BLM P54132 1/20 0.35
PMP22 Q01453 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2958271 0.80 HRH3 (0.59) ALDH1A1KDM4ESMN1; SMN2HRH3CYP1A2
SCHEMBL5221545 0.79 KDM4E (0.65) ALDH1A1KDM4ESMN1; SMN2HRH3CYP1A2
SCHEMBL8765685 0.78 ESR1 (0.41) ESR1ESR2CXCR1ALDH1A1KDM4E
SCHEMBL910859 0.76 NQO1 (0.67) ALDH1A1KDM4ESMN1; SMN2CYP1A2NQO1
SCHEMBL3074697 0.74 KDM4E (0.59) ALDH1A1KDM4ESMN1; SMN2HRH3LTA4H
SCHEMBL24628864 0.74 SLC6A2 (0.44) ESR1ESR2CXCR1ALDH1A1KDM4E
SCHEMBL8765689 0.74 ESR1 (0.59) ESR1ESR2ALDH1A1KDM4ECYP1A2
SCHEMBL8995211 0.73 ALDH1A1 (0.52) ALDH1A1KDM4ESMN1; SMN2HPGD
SCHEMBL6836527 0.73 MMP2 (0.44) ALDH1A1SMN1; SMN2HPGD
SCHEMBL6538461 0.73 SMN1; SMN2 (0.63) ALDH1A1KDM4ESMN1; SMN2KEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5496844-A Indole derivatives OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1996-03-05 US disclosed
EP-0639567-A1 INDOLE DERIVATIVE OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1995-02-22 EP disclosed