SCHEMBL8995535

SCHEMBL8995535

CC(C)(C)OC(=O)C[C@@H](NC(=O)CCc1ccccc1)C(=O)NCCCCc1ccc(C#N)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 7/20 0.46
CTSK P43235 5/20 0.46
GRIA1 P42261 1/20 0.45
CTSB P07858 3/20 0.43
CTSL P07711 2/20 0.43
PTPN1 P18031 1/20 0.43
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA4 P43681 1/20 0.42
NAMPT P43490 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8995530 1.00 CTSS (0.46) CTSSCTSKGRIA1CTSBCTSL
SCHEMBL8995548 0.88 CTSS (0.52) CTSSCTSKCTSBCTSL
SCHEMBL8995562 0.88 CTSS (0.52) CTSSCTSKCTSBCTSL
SCHEMBL7423272 0.88 CTSS (0.52) CTSSCTSKCTSBCTSL
SCHEMBL7421065 0.87 ITGB3 (0.55) GRIA1PTPN1ITGB3ITGA2BCHRNB2
SCHEMBL7421070 0.87 ITGB3 (0.55) GRIA1PTPN1ITGB3ITGA2BCHRNB2
SCHEMBL7417133 0.84 MMP2 (0.50) GRIA1PTPN1ITGB3ITGA2BCHRNB2
SCHEMBL7418533 0.81 CTSS (0.52) CTSSCTSKCTSBCTSLALDH1A1
SCHEMBL8995549 0.81 CTSS (0.52) CTSSCTSKCTSBCTSLALDH1A1
SCHEMBL7423262 0.81 CTSS (0.52) CTSSCTSKCTSBCTSLALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5552431-A ANTICOAGULANTS G. D. SEARLE & CO. (US) 1996-09-03 US disclosed
US-5424334-A Peptide mimetic compounds useful as platelet aggregation inhibitors G. D. SEARLE & CO. (US) 1995-06-13 US disclosed