SCHEMBL8995929

SCHEMBL8995929

C=C1CC(=O)N(c2ccc(Nc3ccc(OC)cc3)cc2)C1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.50
MEN1 O00255 5/20 0.50
KMT2A Q03164 5/20 0.50
RAB9A P51151 3/20 0.50
POLB P06746 1/20 0.50
GAA P10253 7/20 0.48
ALDH1A1 P00352 6/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
RECQL P46063 2/20 0.48
KDM4E B2RXH2 4/20 0.47
TDP1 Q9NUW8 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
NPC1 O15118 2/20 0.47
THRB P10828 1/20 0.47
MAPK1 P28482 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
NR1H2 P55055 1/20 0.46
NR1H3 Q13133 1/20 0.46
APP P05067 1/20 0.45
CYP1A2 P05177 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8995936 0.85 MEN1 (0.55) MAPTMEN1KMT2ARAB9APOLB
SCHEMBL8995982 0.84 MEN1 (0.49) MAPTMEN1KMT2APOLBGAA
SCHEMBL8995947 0.82 HSP90AA1 (0.54) MAPTMEN1KMT2AGAAALDH1A1
SCHEMBL237914 0.78 GAA (0.44) MAPTMEN1KMT2ARAB9APOLB
SCHEMBL30339808 0.75 MAPT (0.61) MAPTMEN1KMT2AGAAALDH1A1
SCHEMBL12220701 0.74 ALDH1A1 (0.62) MAPTMEN1KMT2ARAB9AGAA
SCHEMBL4896862 0.74 GLA (0.63) MAPTMEN1KMT2ARAB9APOLB
SCHEMBL8467713 0.74 MGLL (0.79) MAPTMEN1KMT2ARAB9APOLB
SCHEMBL2983688 0.74 GAA (0.57) MAPTMEN1KMT2ARAB9APOLB
SCHEMBL29250852 0.74 NR1H3 (0.68) MAPTMEN1KMT2ARAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0570825-B1 Tire sidewall composition containing silica having low PH GOODYEAR TIRE & RUBBER (US) 1996-08-07 EP disclosed
EP-0475215-B1 Carboxylic acid esters with thio groups GOODYEAR TIRE & RUBBER (US) 1994-10-19 EP disclosed
EP-0570825-A1 Tire sidewall composition containing silica having low PH THE GOODYEAR TIRE & RUBBER COMPANY (US) 1993-11-24 EP disclosed
US-5244028-A Natural rubber or polybutadiene, silica, antidegradation agent, carbon black THE GOODYEAR TIRE & RUBBER COMPANY (US) 1993-09-14 US disclosed
US-5216049-A A phenolic or amine stabilizer and an organothioalkylene styrene bound to a polymer; aging resistance; rubbers THE GOODYEAR TIRE & RUBBER COMPANY (US) 1993-06-01 US disclosed
EP-0475215-A1 Carboxylic acid esters with thio groups THE GOODYEAR TIRE & RUBBER COMPANY (US) 1992-03-18 EP disclosed
US-5069819-A SYNERGISTS FOR CONVENTIONAL PHENOLIC AND AMINE ANTIOXIDANTS THE GOODYEAR TIRE & RUBBER COMPANY (US) 1991-12-03 US disclosed