SCHEMBL8998849

SCHEMBL8998849

CN1C(=S)Cc2cc(C(F)(F)F)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.43
SCN9A Q15858 1/20 0.39
AADAT Q8N5Z0 1/20 0.38
LMNA P02545 3/20 0.38
POLB P06746 1/20 0.38
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
ALDH1A1 P00352 4/20 0.37
PKM P14618 1/20 0.37
TDP2 O95551 1/20 0.36
BRD4 O60885 1/20 0.36
SRPK1 Q96SB4 1/20 0.36
KDM4E B2RXH2 2/20 0.36
SRD5A1 P18405 1/20 0.35
CA2 P00918 1/20 0.35
KIF11 P52732 1/20 0.35
FPR2 P25090 2/20 0.34
NPC1 O15118 1/20 0.34
MLNR O43193 1/20 0.34
USP1 O94782 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8998844 0.80 LMNA (0.54) NOTUMAADATLMNAPOLBNR1H2
SCHEMBL8999017 0.75 PDE5A (0.39) NOTUMAADATALDH1A1PKMKDM4E
SCHEMBL8998888 0.74 POLB (0.41) NOTUMSCN9AAADATLMNAPOLB
SCHEMBL8999236 0.74 IDO1 (0.38) ALDH1A1TDP2BRD4KDM4ESRD5A1
SCHEMBL16855153 0.73 NR1H2 (0.52) NOTUMSCN9ALMNAPOLBNR1H2
SCHEMBL16817958 0.72 NOTUM (0.49) NOTUMSCN9AAADATNR1H2NR1H3
SCHEMBL8998856 0.71 DRD1 (0.47) NOTUMLMNADRD2DRD1DRD3
SCHEMBL20693639 0.69 NOTUM (0.60) NOTUMSCN9AAADATLMNANR1H2
SCHEMBL8999008 0.69 MAOA (0.40) NOTUMLMNAALDH1A1KDM4ETP53
SCHEMBL12905312 0.67 NOTUM (0.57) NOTUMSCN9AAADATLMNANR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5556874-A ENZYME INHIBITORS AS ANTICARCINOGENIC AGENTS WARNER LAMBERT COMPANY (US) 1996-09-17 US disclosed
US-5464861-A Anticarcinogenic agents WARNER-LAMBERT (US) 1995-11-07 US disclosed
EP-0654024-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1995-05-24 EP disclosed
WO-1994003427-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1994-02-17 WO disclosed