SCHEMBL8999008

SCHEMBL8999008

CN1C(=S)Cc2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.40
HTR2A P28223 3/20 0.40
ADRA2A P08913 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
SLC6A2 P23975 2/20 0.40
HTR2C P28335 2/20 0.40
SLC6A4 P31645 2/20 0.40
ADRA1A P35348 2/20 0.40
HRH1 P35367 2/20 0.40
HTR2B P41595 2/20 0.40
KCNH2 Q12809 2/20 0.40
NOTUM Q6P988 1/20 0.39
DRD2 P14416 2/20 0.39
DRD1 P21728 2/20 0.39
DRD4 P21917 2/20 0.39
DRD3 P35462 2/20 0.39
DRD5 P21918 1/20 0.39
MAPKAPK2 P49137 1/20 0.38
HPGD P15428 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL975897 0.81 MAOA (0.52) MAOAHTR2AADRA2AADRA2BADRA2C
SCHEMBL29351597 0.81 MAOA (0.52) MAOAHTR2AADRA2AADRA2BADRA2C
Iodide SCHEMBL11862710 0.79 MAOA (0.50) MAOAHTR2AADRA2AADRA2BADRA2C
SCHEMBL29735917 0.79 MAOA (0.50) MAOAHTR2AADRA2AADRA2BADRA2C
SCHEMBL3841522 0.79 ALDH1A1 (0.46) HTR2AADRA2BADRA2CSLC6A2HTR2C
SCHEMBL3957285 0.76 ALDH1A1 (0.42) MAOAHTR2AADRA2AADRA2BADRA2C
SCHEMBL9833997 0.75 ADRA2B (0.51) HTR2AADRA2AADRA2BADRA2CSLC6A2
SCHEMBL4442728 0.74 MAOA (0.40) MAOAHTR2AADRA2AADRA2BADRA2C
SCHEMBL12723261 0.74 MAOA (0.45) MAOAHTR2AADRA2AADRA2BADRA2C
SCHEMBL10460338 0.74 CYP1A2 (0.58) MAOAHTR2AADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118048633-A Method for electrochemically synthesizing trifluoro methylthio oxindole 上海电力大学 2024-05-17 CN claimed
CN-118048633-A Method for electrochemically synthesizing trifluoro methylthio oxindole 上海电力大学 2024-05-17 CN disclosed
CN-118048633-A Method for electrochemically synthesizing trifluoro methylthio oxindole 上海电力大学 2024-05-17 CN disclosed
CN-118048633-A Method for electrochemically synthesizing trifluoro methylthio oxindole 上海电力大学 2024-05-17 CN disclosed
US-5556874-A ENZYME INHIBITORS AS ANTICARCINOGENIC AGENTS WARNER LAMBERT COMPANY (US) 1996-09-17 US disclosed
US-5464861-A Anticarcinogenic agents WARNER-LAMBERT (US) 1995-11-07 US disclosed
EP-0654024-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1995-05-24 EP disclosed
WO-1994003427-A1 2-THIOINDOLES (SELENOINDOLES) AND RELATED DISULFIDES (SELENIDES) WHICH INHIBIT PROTEIN TYROSINE KINASES AND WHICH HAVE ANTITUMOR PROPERTIES WARNER-LAMBERT COMPANY (US) 1994-02-17 WO disclosed
US-5030646-A Treatment of diseases resulting from disfunction of seretoninergic system ADIR ET COMPAGNIE (FR) 1991-07-09 US disclosed