SCHEMBL9002406

SCHEMBL9002406

O=C(c1cccnc1-c1cc([N+](=O)[O-])cc(C(F)(F)F)c1)c1cccnc1-c1cc([N+](=O)[O-])cc(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.44
P2RX1 P51575 5/20 0.43
TP53 P04637 1/20 0.41
RORB Q92753 3/20 0.40
PDE4D Q08499 1/20 0.40
P2RX4 Q99571 1/20 0.39
P2RX7 Q99572 1/20 0.39
MAPT P10636 4/20 0.39
HTT P42858 2/20 0.39
LMNA P02545 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
NFKB1 P19838 1/20 0.39
CASP6 P55212 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002865 0.79 PDE4D (0.61) RORBPDE4DMAPTNPC1RAB9A
SCHEMBL9002267 0.78 RORB (0.56) TRPV1RORBLMNATDP1PKM
SCHEMBL9002089 0.75 NR2E1 (0.46) TRPV1P2RX1RORBP2RX4P2RX7
SCHEMBL10768030 0.70 PDE4D (0.60) TP53PDE4DMAPTNPC1RAB9A
SCHEMBL7273341 0.70 PDE4D (0.60) TP53PDE4DMAPTNPC1RAB9A
SCHEMBL27993567 0.69 KMT2A (0.60) PDE4DMAPTNPC1RAB9ATDP1
SCHEMBL9002388 0.69 GPBAR1 (0.52) MAPTHTTLMNAGPBAR1MEN1
SCHEMBL30600332 0.69 CYP19A1 (0.64) P2RX1MAPTLMNATDP1SCN2A
SCHEMBL473595 0.69 ALDH1A1 (0.59) TRPV1RORBLMNARAB9ATDP1
SCHEMBL29319717 0.68 CYP19A1 (0.48) P2RX1P2RX4P2RX7HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5482948-A Pyridyl derivatives and pharmaceutical compositions comprising these compounds DR. KARL THOMAE GMBH (DE) 1996-01-09 US disclosed