SCHEMBL9005979

SCHEMBL9005979

Cc1cc2nc(CCC(=O)O)c(CP(=O)(O)O)c(N)c2cc1C

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PGK1 P00558 1/20 0.36
PGK2 P07205 1/20 0.36
HDAC6 Q9UBN7 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
DPP4 P27487 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9005973 0.68 BCAT2 (0.38) HDAC6L3MBTL1NPSR1
SCHEMBL8645093 0.67 PRKAG1 (0.37) PGK1PGK2NPSR1
SCHEMBL9700784 0.63 HDAC6 (0.41) KDM4EHSD17B10PGK1PGK2HDAC6
SCHEMBL9741731 0.63
SCHEMBL6666177 0.63 EGFR (0.49) KDM4EHSD17B10
SCHEMBL28453316 0.61 SLC22A12 (0.38) KDM4EHDAC6L3MBTL1NPSR1
SCHEMBL28447347 0.61 GAA (0.36) KDM4EHSD17B10HDAC6L3MBTL1NPSR1
SCHEMBL8644134 0.60
SCHEMBL9701703 0.59 PLAU (0.34)
SCHEMBL9742575 0.59

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0736032-A1 HETEROCYCLIC COMPOUNDS Astra Aktiebolag (SE) 1996-10-09 EP disclosed
WO-1995017410-A1 HETEROCYCLIC COMPOUNDS ASTRA AKTIEBOLAG (SE) 1995-06-29 WO disclosed