SCHEMBL9007535

SCHEMBL9007535

COC(=O)NC(=O)CC1=C(Cc2ccc3c(Cl)cccc3c2)C(=O)CC1

nearest known ligand 0.32

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LDHA P00338 2/20 0.32
TSHR P16473 1/20 0.32
TRPV1 Q8NER1 1/20 0.31
ATM Q13315 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
S1PR1 P21453 1/20 0.31
CRHBP P24387 1/20 0.31
CRHR2 Q13324 1/20 0.31
KDM4E B2RXH2 2/20 0.30
ALDH1A1 P00352 2/20 0.30
HPGD P15428 1/20 0.30
POLB P06746 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
AKR1B1 P15121 1/20 0.30
NQO2 P16083 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9007576 0.83 MEN1 (0.32) ATMMEN1KMT2AALDH1A1HPGD
SCHEMBL9007566 0.83 AKR1B1 (0.42) LDHAAKR1B1
SCHEMBL9007525 0.78 AKR1B1 (0.41) LDHAAKR1B1
SCHEMBL9007582 0.72 KMT2A (0.40) TSHRKMT2AKDM4EALDH1A1HPGD
SCHEMBL9007553 0.72 NQO1 (0.37) MEN1KMT2AALDH1A1POLBCYP3A4
SCHEMBL9007515 0.69 KMT2A (0.39) TSHRKMT2AKDM4EALDH1A1HPGD
SCHEMBL9007517 0.65 AKR1B1 (0.41) MEN1KMT2AKDM4EPOLBAKR1B1
SCHEMBL11740657 0.64 AKR1B1 (0.60) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL15715945 0.62 CYP1A2 (0.44) MEN1KMT2AALDH1A1CYP3A4CYP2C9
SCHEMBL9007552 0.62 GAA (0.40) TSHRKMT2AKDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5482968-A ENZYME INHIBITORS, HYPOGLYCEMIC AGENTS AND VASCULAR AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1996-01-09 US claimed
US-5399588-A Diabetes treatment AMERICAN HOME PRODUCTS CORPORATION (US) 1995-03-21 US claimed
US-5482968-A ENZYME INHIBITORS, HYPOGLYCEMIC AGENTS AND VASCULAR AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1996-01-09 US disclosed
US-5399588-A Diabetes treatment AMERICAN HOME PRODUCTS CORPORATION (US) 1995-03-21 US disclosed