SCHEMBL9010704

SCHEMBL9010704

NC(=S)Nc1cccc(B(O)O)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.59
CYP1A2 P05177 1/20 0.58
ALDH1A1 P00352 3/20 0.53
TP53 P04637 1/20 0.53
TYR P14679 1/20 0.53
TSHR P16473 1/20 0.53
TAS2R38 P59533 1/20 0.53
HSD17B10 Q99714 1/20 0.53
ENPP2 Q13822 2/20 0.47
KDM4E B2RXH2 2/20 0.47
TRPV1 Q8NER1 1/20 0.44
NLRP3 Q96P20 1/20 0.44
RXFP1 Q9HBX9 1/20 0.42
IDO1 P14902 1/20 0.42
ESRRG P62508 2/20 0.42
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
MGLL Q99685 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13715294 0.85 TAS2R38 (0.53) KMT2ACYP1A2ALDH1A1TAS2R38ENPP2
SCHEMBL4047674 0.82 KMT2A (0.76) KMT2ACYP1A2ALDH1A1TP53TYR
SCHEMBL1303751 0.81 TRPV1 (0.51) ALDH1A1ENPP2KDM4ETRPV1NLRP3
SCHEMBL10712920 0.81 ENPP2 (0.47) KMT2AALDH1A1ENPP2KDM4ETRPV1
SCHEMBL6357941 0.80 ALDH1A1 (0.61) KMT2ACYP1A2ALDH1A1TAS2R38HSD17B10
SCHEMBL2554968 0.79 ALDH1A1 (0.57) KMT2ACYP1A2ALDH1A1KDM4ETRPV1
SCHEMBL147446 0.77 IDO1 (0.68) KMT2ACYP1A2ALDH1A1TP53TYR
SCHEMBL29838519 0.77 IDO1 (0.68) KMT2ACYP1A2ALDH1A1TP53TYR
SCHEMBL2564353 0.76 TRPV1 (0.52) ALDH1A1ENPP2KDM4ETRPV1NLRP3
SCHEMBL2559389 0.75 KDM4E (0.48) ALDH1A1KDM4ETRPV1NLRP3IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0279307-B2 Bifunctional chelating agents ABBOTT LAB (US) 1996-11-13 EP disclosed
EP-0315188-B1 Methods and materials for the preparation of metal labelled antibody solutions ABBOTT LAB (US) 1994-06-01 EP disclosed
US-5245026-A Radiopharmaceutical applications ABBOTT LABORATORIES (US) 1993-09-14 US disclosed
US-5227474-A Complexing with radioactive metals, binding to biologically active molecules for treatment of tumors and diagnostic imaging ABBOTT LABORATORIES (US) 1993-07-13 US disclosed
EP-0308757-B1 MULTIDENTATE CHELATORS BASED ON THE 8-HYDROXYQUINOLINE UNIT ABBOTT LABORATORIES (US) 1993-06-30 EP disclosed
US-5217704-A Methods and materials for the preparation of metal labelled antibody solutions ABBOTT LABORATORIES (US) 1993-06-08 US disclosed
US-5130118-A Radioactive metal ion labelled chelator ABBOTT LABORATORIES (US) 1992-07-14 US disclosed
US-5057302-A Stable metal complexes of a substrate having a carboxymethyl arm of a polyaminopolycarboxylate framework; medical diagnosis; immunoassay; radiology; antitumor and anticarcinogenic agents ABBOTT LABORATORIES (US) 1991-10-15 US disclosed
US-5021567-A Medical diagnosis; radiology; immunology; demetallization; stable complexes ABBOTT LABORATORIES (US) 1991-06-04 US disclosed
EP-0315188-A2 Methods and materials for the preparation of metal labelled antibody solutions ABBOTT LABORATORIES (US) 1989-05-10 EP disclosed
EP-0308757-A1 Multidentate chelators based on the 8-hydroxyquinoline unit ABBOTT LABORATORIES (US) 1989-03-29 EP disclosed
EP-0279307-A2 Bifunctional chelating agents ABBOTT LABORATORIES (US) 1988-08-24 EP disclosed