SCHEMBL9010784

SCHEMBL9010784

CC(C)(NC(=O)c1cncc(Cl)c1)C(=O)C(Br)Br

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.45
USP36 Q9P275 1/20 0.43
SMYD3 Q9H7B4 1/20 0.42
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
NTRK1 P04629 1/20 0.35
EGFR P00533 1/20 0.35
CNR2 P34972 1/20 0.35
S1PR4 O95977 1/20 0.35
S1PR3 Q99500 1/20 0.35
KDM4E B2RXH2 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KCNH2 Q12809 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
ACKR3 P25106 1/20 0.33
DDR1 Q08345 1/20 0.33
KMT2A Q03164 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8400032 0.84 GRN (0.46) KCNH2KMT2A
SCHEMBL8402049 0.79 GPR139 (0.42) DDR1KMT2A
SCHEMBL8403842 0.78 TAS1R3 (0.46) SLC6A3KCNH2DDR1TAS1R3TAS1R1
SCHEMBL8402078 0.78 GRN (0.38) CNR2KCNH2KMT2A
SCHEMBL9010830 0.76 HDAC1 (0.51) KMT2A
SCHEMBL9821286 0.75 RAB9A (0.48) EGFRKMT2A
SCHEMBL9082843 0.75 HPGD (0.48) PTGS2KDM4ETAS1R3TAS1R1TAS1R2
SCHEMBL8400028 0.74 HPGD (0.49) KDM4EKMT2ATAS1R3TAS1R2
SCHEMBL8403929 0.74 GRN (0.44) KCNH2KMT2A
SCHEMBL8402033 0.73 LMNA (0.35) KDM4EDDR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5547984-A FUNGICIDES ROHM AND HAAS COMPANY (US) 1996-08-20 US disclosed
US-5529978-A FUNGICIDE ROHM AND HAAS COMPANY (US) 1996-06-25 US disclosed
US-5344978-A Fungicides ROHM AND HAAS COMPANY (US) 1994-09-06 US disclosed
US-5196046-A N-acetonyl-substituted-amides ROHM AND HAAS COMPANY (US) 1993-03-23 US disclosed
EP-0170498-B1 N-ACETONYL-SUBSTITUTED-AMIDES, COMPOSITIONS CONTAINING THEM AND THEIR USE IN COMBATING FUNGI ROHM AND HAAS COMPANY (US) 1991-09-11 EP disclosed
US-4863940-A N-acetonyl-substituted amides and phytopathogenic fungicidal use thereof ROHM AND HAAS (US) 1989-09-05 US disclosed
EP-0170498-A2 N-acetonyl-substituted-amides, compositions containing them and their use in combating fungi ROHM AND HAAS COMPANY (US) 1986-02-05 EP disclosed