SCHEMBL901121

SCHEMBL901121

[CH2]Cc1ccc(Cl)c(Cl)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.40
MAPK1 P28482 1/20 0.40
PNMT P11086 1/20 0.36
AHR P35869 2/20 0.34
TDP1 Q9NUW8 1/20 0.33
TAAR1 Q96RJ0 1/20 0.32
IDO1 P14902 3/20 0.31
CYP2A6 P11509 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4465598 0.78 CYP3A4 (0.43) CYP3A4MAPK1PNMTAHRTDP1
SCHEMBL1547863 0.77 PNMT (0.62) CYP3A4PNMTTAAR1IDO1CYP2A6
SCHEMBL12474340 0.77 TAAR1 (0.36) CYP3A4MAPK1PNMTAHRTAAR1
SCHEMBL3727971 0.76 CYP3A4 (0.42) CYP3A4MAPK1PNMTAHRTDP1
SCHEMBL10414261 0.75 TAAR1 (0.35) CYP3A4MAPK1PNMTTAAR1
SCHEMBL5003742 0.75 PNMT (0.43) PNMTTAAR1IDO1
SCHEMBL2090168 0.74 CYP3A4 (0.46) CYP3A4MAPK1PNMTAHRTDP1
SCHEMBL2095375 0.74 PNMT (0.65) CYP3A4MAPK1PNMTAHRTDP1
SCHEMBL2090165 0.74 CYP3A4 (0.40) CYP3A4MAPK1PNMTAHRTDP1
SCHEMBL6305999 0.74 CYP3A4 (0.40) CYP3A4MAPK1PNMTAHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2621922-A1 A PROCESS FOR THE SYNTHESIS OF THIO-TRIAZOLO-GROUP CONTAINING COMPOUNDS BASF SE (DE) 2013-08-07 EP disclosed
US-8426631-B2 Fungicidal compounds, method for the production thereof, and use thereof to combat damaging fungi, and agents comprising the same BASF SE (DE) 2013-04-23 US disclosed
WO-2012041858-A1 A PROCESS FOR THE SYNTHESIS OF THIO-TRIAZOLO-GROUP CONTAINING COMPOUNDS BASF SE (DE) 2012-04-05 WO disclosed
EP-2311816-A1 Isoxazoline Compounds and their Use in Pest Control Sumitomo Chemical Company, Limited (JP) 2011-04-20 EP disclosed
EP-2311817-A1 Isoxazoline Compounds and their Use in Pest Control Sumitomo Chemical Company, Limited (JP) 2011-04-20 EP disclosed
EP-2308858-A1 Isoxazoline Compounds and their Use in Pest Control Sumitomo Chemical Company, Limited (JP) 2011-04-13 EP disclosed
US-20100304966-A1 Fungicidal Compounds, Method For the Production Thereof, And Use Thereof To Combat Damaging Fungi, And Agents Comprising The Same BASF SE (DE) 2010-12-02 US disclosed
US-20100137372-A1 ISOXAZOLINE COMPOUNDS AND THEIR USE IN PEST CONTROL SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2010-06-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137372-A1 ISOXAZOLINE COMPOUNDS AND THEIR USE IN PEST CONTROL CYP4X1, PRDX5, PRDX1 CYP3A4 95/4885MAPK1 3232/4885PNMT 494/4885
US-20100304966-A1 Fungicidal Compounds, Method For the Production Thereof, And Use Thereof To Combat Damaging Fungi, And Agents Comprising The Same CYP51A1, ERG28, CAT CYP3A4 55/4885MAPK1 1845/4885PNMT 591/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.