SCHEMBL9014137

SCHEMBL9014137

CCCCCCN(C(C)=O)c1ccc(OC2CCNCC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 3/20 0.40
NPC1 O15118 1/20 0.39
JAK2 O60674 1/20 0.39
RAB9A P51151 1/20 0.39
PAX8 Q06710 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
GNAI3 P08754 1/20 0.37
GNAO1 P09471 1/20 0.37
GNAI1 P63096 1/20 0.37
GRK6 P43250 1/20 0.37
HRH3 Q9Y5N1 2/20 0.37
MLYCD O95822 3/20 0.36
ACHE P22303 1/20 0.36
CFTR P13569 1/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
OPRM1 P35372 1/20 0.35
MLNR O43193 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014145 0.80 HRH1 (0.42) HRH1NPC1JAK2RAB9APAX8
SCHEMBL9013995 0.79 GPR119 (0.51)
SCHEMBL9014111 0.79 ACHE (0.61) HRH3ACHEOPRM1
SCHEMBL3930753 0.74 NPC1 (0.50) NPC1JAK2RAB9APAX8CHRM2
SCHEMBL13791513 0.72 NPC1 (0.55) NPC1JAK2RAB9APAX8MLYCD
SCHEMBL13791624 0.72 NPC1 (0.48) NPC1JAK2RAB9APAX8CHRM2
SCHEMBL8390888 0.72 NPC1 (0.51) NPC1JAK2RAB9APAX8CHRM2
SCHEMBL9014140 0.72 HRH1 (0.54) HRH1GNAI3GNAO1GNAI1
SCHEMBL13791114 0.71 RAB9A (0.53) NPC1JAK2RAB9APAX8MLYCD
SCHEMBL9809230 0.71 NPC1 (0.69) NPC1JAK2RAB9APAX8CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5580883-A INHIBITING DEGENERATION AND NECROCYTOSIS OF CEREBRAL NERVE CELLS CAUSED BY OXIDATIVE STRESS INDUCING GLUTAMIC ACID IN MAMMALS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-03 US disclosed
EP-0449195-B1 Aminobenzene compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-05-08 EP disclosed
EP-0449195-A2 Aminobenzene compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-10-02 EP disclosed