SCHEMBL9014337

SCHEMBL9014337

CC(=O)Nc1cccc2c1C(CCBr)CCCO2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 0.42
MTNR1B P49286 4/20 0.42
CASP1 P29466 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HSD17B10 Q99714 2/20 0.36
ALOX15 P16050 1/20 0.36
MAP3K14 Q99558 1/20 0.35
LMNA P02545 2/20 0.34
RAB9A P51151 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ADRA2A P08913 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014383 0.80 MTNR1A (0.40) MTNR1AMTNR1BMAP3K14L3MBTL1
SCHEMBL9014723 0.76 MAP3K14 (0.36) MTNR1AMTNR1BMAP3K14
SCHEMBL9014396 0.75 MAP3K14 (0.35) MTNR1AMTNR1BMAP3K14
SCHEMBL9015271 0.75 MAP3K14 (0.35) MTNR1AMTNR1BMAP3K14
SCHEMBL9014644 0.74 KCNH2 (0.59)
SCHEMBL9014349 0.72 CHRNB4 (0.36) ALDH1A1MAP3K14RAB9AL3MBTL1MEN1
SCHEMBL9014726 0.72 MAP3K14 (0.33) MTNR1AMTNR1BMAP3K14RAB9AKMT2A
SCHEMBL9014727 0.69 KCNH2 (0.38) MTNR1AMTNR1BLMNA
SCHEMBL2961606 0.67 MTNR1A (0.57) MTNR1ACASP1KDM4EALDH1A1HSD17B10
SCHEMBL10813137 0.66 MTNR1B (0.55) MTNR1AMTNR1BCASP1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed