SCHEMBL9014396

SCHEMBL9014396

Nc1cccc2c1C(CCBr)CCCO2

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 1/20 0.35
MTNR1A P48039 1/20 0.31
MTNR1B P49286 1/20 0.31
CHRNB4 P30926 2/20 0.30
CHRNA3 P32297 2/20 0.30
CHRNB2 P17787 1/20 0.30
CHRNA4 P43681 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014723 0.84 MAP3K14 (0.36) MAP3K14MTNR1AMTNR1B
SCHEMBL9015271 0.83 MAP3K14 (0.35) MAP3K14MTNR1AMTNR1B
SCHEMBL9014787 0.80 HTR1A (0.39) MAP3K14
SCHEMBL9014726 0.80 MAP3K14 (0.33) MAP3K14MTNR1AMTNR1B
SCHEMBL9014349 0.78 CHRNB4 (0.36) MAP3K14CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL9014727 0.76 KCNH2 (0.38) MTNR1AMTNR1B
SCHEMBL9014383 0.76 MTNR1A (0.40) MAP3K14MTNR1AMTNR1B
SCHEMBL9014337 0.75 MTNR1A (0.42) MAP3K14MTNR1AMTNR1B
SCHEMBL9014335 0.71 KDM4E (0.37) MTNR1AMTNR1BCHRNB4CHRNA3CHRNB2
SCHEMBL9772853 0.66 KCNH2 (0.44) MAP3K14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed