SCHEMBL9014349

SCHEMBL9014349

O=[N+]([O-])c1cccc2c1C(CCBr)CCCO2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 2/20 0.36
CHRNA3 P32297 2/20 0.36
ALDH1A1 P00352 4/20 0.34
HPGD P15428 1/20 0.34
ACHE P22303 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
MAPT P10636 2/20 0.32
NPC1 O15118 2/20 0.32
S1PR4 O95977 1/20 0.32
S1PR1 P21453 1/20 0.32
TDP1 Q9NUW8 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MAP3K14 Q99558 1/20 0.31
S100A4 P26447 1/20 0.31
HCAR3 P49019 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014723 0.79 MAP3K14 (0.36) MAP3K14
SCHEMBL9015271 0.78 MAP3K14 (0.35) SMN1; SMN2MAP3K14
SCHEMBL9014396 0.78 MAP3K14 (0.35) CHRNB4CHRNA3CHRNB2CHRNA4MAP3K14
SCHEMBL9014643 0.75 TERT (0.38) CHRNB4CHRNA3ALDH1A1ACHEMEN1
SCHEMBL9014787 0.74 HTR1A (0.39) MAP3K14
SCHEMBL9014726 0.74 MAP3K14 (0.33) KMT2ANPC1TDP1MAP3K14RAB9A
SCHEMBL9014337 0.72 MTNR1A (0.42) ALDH1A1L3MBTL1MEN1KMT2ATDP1
SCHEMBL9014727 0.71 KCNH2 (0.38) SMN1; SMN2
SCHEMBL5839690 0.66 MAPT (0.43) CHRNB4CHRNA3ALDH1A1HPGDMAPT
SCHEMBL10407545 0.64 HSP90AA1 (0.38) CHRNB4CHRNA3ALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5495022-A Piperidines and piperazines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-02-27 US disclosed
EP-0634398-A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents MERCK PATENT GmbH (DE) 1995-01-18 EP disclosed