SCHEMBL9014886

SCHEMBL9014886

Clc1cccnc1N1CCN(CCCCOc2cnc3c(n2)CCCC3)CC1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 4/20 0.46
KCNH2 Q12809 3/20 0.46
HTR1A P08908 7/20 0.43
DRD2 P14416 7/20 0.43
HTR2A P28223 7/20 0.43
HTR7 P34969 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
DRD1 P21728 1/20 0.41
DRD4 P21917 1/20 0.41
DRD5 P21918 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
ADRA1A P35348 1/20 0.40
HRH1 P35367 1/20 0.40
ADRA1B P35368 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014877 0.86 DRD2 (0.52) DRD3HTR1ADRD2HTR2AHTR7
SCHEMBL9014712 0.85 DRD2 (0.57) HTR1ADRD2HTR2AHTR7DRD4
SCHEMBL9014896 0.85 HSD11B1 (0.49) HTR1ADRD2HTR2A
SCHEMBL9014893 0.83 HRH3 (0.50) DRD3KCNH2HTR1ADRD2HTR2A
SCHEMBL9014651 0.83 HTR1A (0.43) HTR1ADRD2HTR2AHRH3
SCHEMBL9014904 0.82 HRH3 (0.49) DRD3KCNH2HTR1ADRD2HTR2A
SCHEMBL9014815 0.82 KCNH2 (0.55) DRD3KCNH2HTR1ADRD2HTR2A
SCHEMBL9014858 0.81 KCNH2 (0.57) DRD3KCNH2HTR1ADRD2HTR2A
SCHEMBL9014870 0.80 HTR3E (0.45) DRD3KCNH2HTR1ADRD2HTR2A
SCHEMBL9014894 0.80 DRD2 (0.52) DRD3KCNH2HTR1ADRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5578596-A TREATMENT OF SEROTONERGIC NEURON RELATED DISEASES, MOTION SICKNESS, ANXIXETY, DEPRESSION ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1996-11-26 US disclosed
EP-0668276-A1 2-ALKOXY-5,6,7,8-TETRAHYDROQUINOXALINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1995-08-23 EP disclosed