SCHEMBL9017918

SCHEMBL9017918

CN(C)C(=O)Oc1cnccc1N=CN(C)C1CCCCC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.34
NCEH1 Q6PIU2 2/20 0.33
ACHE P22303 5/20 0.33
PRMT3 O60678 1/20 0.33
ALDH1A1 P00352 2/20 0.33
POLB P06746 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
GAA P10253 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
LCK P06239 1/20 0.32
JAK3 P52333 1/20 0.32
OPRK1 P41145 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL9017934 0.95 BCHE (0.31) BCHENCEH1ACHEPRMT3ALDH1A1
Fumaric Acid SCHEMBL9017938 0.95 BCHE (0.31) BCHENCEH1ACHEPRMT3ALDH1A1
SCHEMBL9017936 0.89 MEN1 (0.30) ALDH1A1MAPK1
SCHEMBL9017843 0.82 RAB9A (0.38) BCHENCEH1ALDH1A1TSHRGAA
SCHEMBL9017846 0.82 RAB9A (0.38) BCHENCEH1ALDH1A1TSHRGAA
SCHEMBL9017879 0.79 ACHE (0.39) BCHENCEH1ACHETSHR
SCHEMBL9017892 0.79 ACHE (0.39) BCHENCEH1ACHETSHR
SCHEMBL9017889 0.79 ACHE (0.39) BCHENCEH1ACHETSHR
SCHEMBL9017875 0.79 ACHE (0.39) BCHENCEH1ACHETSHR
SCHEMBL9017858 0.78 CACNA1B (0.34) PRMT3ALDH1A1POLBTSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0477903-B1 Substituted-4-amino-3-pyridinols, a process for their preparation and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1996-04-03 EP disclosed
EP-0477903-A2 Substituted-4-amino-3-pyridinols, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-04-01 EP disclosed