SCHEMBL9018007

SCHEMBL9018007

COC(=O)Oc1ccc(C(=O)NS(=O)(=O)c2cccc(C(=O)NCCCCc3ccccc3)c2)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
TP53 P04637 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HPGD P15428 4/20 0.45
KDM4E B2RXH2 3/20 0.45
MAPT P10636 3/20 0.45
CYP2D6 P10635 6/20 0.44
CYP2C9 P11712 6/20 0.44
CYP1A2 P05177 4/20 0.44
CYP2C19 P33261 3/20 0.44
MYOF Q9NZM1 2/20 0.44
GLA P06280 1/20 0.43
EPHX2 P34913 1/20 0.43
P4HTM Q9NXG6 1/20 0.43
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9018085 0.97 RAB9A (0.47) ALDH1A1RAB9ASMN1; SMN2NPC1TP53
SCHEMBL9018282 0.94 RAB9A (0.53) ALDH1A1RAB9ASMN1; SMN2NPC1TP53
SCHEMBL9018465 0.93 ALDH1A1 (0.44) ALDH1A1RAB9ASMN1; SMN2NPC1TP53
SCHEMBL9018093 0.92 ALDH1A1 (0.42) ALDH1A1RAB9ASMN1; SMN2NPC1TP53
SCHEMBL9018225 0.91 HSP90AA1 (0.47) ALDH1A1RAB9ASMN1; SMN2NPC1HPGD
SCHEMBL9018010 0.91 RAB9A (0.44) ALDH1A1RAB9ASMN1; SMN2NPC1TP53
SCHEMBL9018274 0.90 RAB9A (0.48) ALDH1A1RAB9ASMN1; SMN2NPC1TP53
SCHEMBL9018042 0.90 SMN1; SMN2 (0.43) SMN1; SMN2HDAC6MAPTP4HTMHTT
SCHEMBL9018296 0.89 HTT (0.55) ALDH1A1RAB9AHDAC2HDAC8HDAC6
SCHEMBL9018092 0.89 SMN1; SMN2 (0.47) ALDH1A1RAB9ASMN1; SMN2MAPTGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0590520-B1 Acylsulphonamido and sulphonamidopyridine-2-carboxylic acid esters, pyridine-n-oxides thereof, a process for their preparation and their use as medicaments HOECHST AG (DE) 1996-06-12 EP disclosed
EP-0590520-A1 Acylsulphonamido and sulphonamidopyridine-2-carboxylic acid esters, pyridine-n-oxides thereof, a process for their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1994-04-06 EP disclosed