SCHEMBL9018062

SCHEMBL9018062

O=C(Oc1ccc(C(=O)NS(=O)(=O)c2ccc(C(=O)NCCc3ccccc3)cc2)cn1)OC1CCCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.45
NPC1 O15118 5/20 0.45
RAB9A P51151 5/20 0.45
MAPT P10636 4/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 2/20 0.44
TSHR P16473 2/20 0.44
KDM4E B2RXH2 1/20 0.44
TP53 P04637 1/20 0.44
HPGD P15428 1/20 0.44
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
P4HTM Q9NXG6 2/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
CYP3A4 P08684 1/20 0.42
HTR1A P08908 1/20 0.42
CYP2C9 P11712 1/20 0.42
NFKB1 P19838 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9018210 0.99 SMN1; SMN2 (0.45) SMN1; SMN2NPC1RAB9AMAPTALDH1A1
SCHEMBL9018058 0.94 ACACB (0.43) SMN1; SMN2NPC1RAB9AALDH1A1HTT
SCHEMBL9018508 0.93 HSP90AA1 (0.42) NPC1RAB9AALDH1A1HTTNPSR1
SCHEMBL9018079 0.92 ALDH1A1 (0.42) SMN1; SMN2RAB9AMAPTALDH1A1LMNA
SCHEMBL9018393 0.92 CXCR1 (0.47) SMN1; SMN2NPC1RAB9AMAPTLMNA
SCHEMBL9018083 0.91 SCN3A (0.46) SMN1; SMN2RAB9AMAPTALDH1A1LMNA
SCHEMBL9018390 0.91 CA1 (0.44) SMN1; SMN2NPC1RAB9AMAPTALDH1A1
SCHEMBL9018073 0.91 EGFR (0.46) SMN1; SMN2NPC1RAB9AMAPTALDH1A1
SCHEMBL9018540 0.90 RAB9A (0.47) SMN1; SMN2NPC1RAB9AALDH1A1HPGD
SCHEMBL9018159 0.89 KMT2A (0.49) SMN1; SMN2NPC1RAB9AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0590520-B1 Acylsulphonamido and sulphonamidopyridine-2-carboxylic acid esters, pyridine-n-oxides thereof, a process for their preparation and their use as medicaments HOECHST AG (DE) 1996-06-12 EP disclosed
EP-0590520-A1 Acylsulphonamido and sulphonamidopyridine-2-carboxylic acid esters, pyridine-n-oxides thereof, a process for their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1994-04-06 EP disclosed