SCHEMBL9018250

SCHEMBL9018250

CCC(CC)OC(=O)Oc1ccc(C(=O)NS(=O)(=O)c2cccc(CCNC(=O)CC3CCCCC3)c2)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.43
ALDH1A1 P00352 1/20 0.36
PKM P14618 1/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
OPRM1 P35372 2/20 0.35
OPRD1 P41143 2/20 0.35
OPRK1 P41145 1/20 0.35
LMNA P02545 1/20 0.35
CYP3A4 P08684 1/20 0.35
HTR1A P08908 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
NFKB1 P19838 1/20 0.35
CNR1 P21554 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9018312 0.93 EPHX2 (0.47) EPHX2ALDH1A1PKMOPRM1OPRD1
SCHEMBL9018486 0.92 LMNA (0.42) EPHX2ALDH1A1OPRM1OPRD1OPRK1
SCHEMBL9018191 0.90 EPHX2 (0.41) EPHX2ALDH1A1PKMCA1CA2
SCHEMBL9018252 0.90 MEN1 (0.39) ALDH1A1LMNACYP3A4HTR1AMAPT
SCHEMBL9018435 0.87 ALDH1A1 (0.39) ALDH1A1CA1CA2CA7CA9
SCHEMBL9018301 0.87 CA1 (0.41) ALDH1A1CA1CA2CA7CA9
SCHEMBL9018198 0.87 OPRM1 (0.40) ALDH1A1CA1CA2CA7CA9
SCHEMBL9018345 0.87 OPRM1 (0.40) EPHX2ALDH1A1CA1CA2CA7
SCHEMBL7862673 0.85 EPHX2 (0.44) EPHX2ALDH1A1PKMLMNACYP3A4
SCHEMBL7867707 0.85 EPHX2 (0.46) EPHX2ALDH1A1PKMLMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0590520-B1 Acylsulphonamido and sulphonamidopyridine-2-carboxylic acid esters, pyridine-n-oxides thereof, a process for their preparation and their use as medicaments HOECHST AG (DE) 1996-06-12 EP disclosed
EP-0590520-A1 Acylsulphonamido and sulphonamidopyridine-2-carboxylic acid esters, pyridine-n-oxides thereof, a process for their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1994-04-06 EP disclosed