SCHEMBL9018719

SCHEMBL9018719

NC(N)=NC(=O)c1cc(C(F)(F)F)ccc1[N+](=O)[O-]

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.46
AKR1C4 P17516 1/20 0.46
AKR1C3 P42330 1/20 0.46
AKR1C2 P52895 1/20 0.46
AKR1C1 Q04828 1/20 0.46
TTR P02766 2/20 0.46
MEN1 O00255 1/20 0.46
PPOX P50336 1/20 0.46
KMT2A Q03164 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
MAPT P10636 3/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HPD P32754 3/20 0.44
SLC9A1 P19634 3/20 0.43
P2RX1 P51575 1/20 0.43
KCNMA1 Q12791 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8612597 0.91 CFTR (0.48) AKR1B1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL28865598 0.84 AKR1B1 (0.51) AKR1B1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL9018718 0.80 SLC9A1 (0.41) TTRMEN1PPOXKMT2ATDP1
SCHEMBL16031334 0.79 TTR (0.64) AKR1B1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL9018707 0.78 SLC9A1 (0.46) SLC9A1ALDH1A1PLAU
SCHEMBL9018662 0.78 CES2 (0.62) SLC9A1ALDH1A1PLAU
SCHEMBL16620136 0.77 TDP1 (0.47) AKR1B1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL9018705 0.77 SLC9A1 (0.48) SLC9A1PLAU
Hydrochloric Acid SCHEMBL8393445 0.77 SLC9A1 (0.45) SLC9A1ALDH1A1PLAU
Hydrochloric Acid SCHEMBL8393438 0.77 CES2 (0.60) SLC9A1ALDH1A1PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743301-A2 Benzoylguanidines containing fluorine MERCK PATENT GmbH (DE) 1996-11-20 EP disclosed