SCHEMBL9019339

SCHEMBL9019339

CCCCCCCCCCCCCCCCSCc1c(-c2ccc(OC)cc2)oc2cc(O)cc(O)c2c1=O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.60
ABCB1 P08183 3/20 0.60
CYP1B1 Q16678 3/20 0.60
CYP1A1 P04798 2/20 0.60
CYP1A2 P05177 2/20 0.60
FTO Q9C0B1 1/20 0.60
CYP3A4 P08684 4/20 0.59
CYP2D6 P10635 4/20 0.59
POLH Q9Y253 4/20 0.52
KDM4E B2RXH2 3/20 0.50
RECQL P46063 3/20 0.50
POLB P06746 2/20 0.50
APEX1 P27695 2/20 0.50
MCL1 Q07820 1/20 0.50
GLO1 Q04760 1/20 0.49
MEN1 O00255 3/20 0.47
MAPT P10636 3/20 0.47
KMT2A Q03164 3/20 0.47
NPC1 O15118 2/20 0.47
ALDH1A1 P00352 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9019366 0.76 CYP19A1 (0.56) MAOAABCB1CYP1B1CYP1A1CYP1A2
Kaempferide SCHEMBL426774 0.76 CYP1A2 (1.00) MAOAABCB1CYP1B1CYP1A1CYP1A2
Kaempferide SCHEMBL29371282 0.76 CYP1A2 (1.00) MAOAABCB1CYP1B1CYP1A1CYP1A2
Ermanin SCHEMBL2875089 0.75 CYP3A4 (1.00) MAOAABCB1CYP1B1CYP1A1CYP1A2
SCHEMBL6504199 0.74 CYP1B1 (0.77) MAOAABCB1CYP1B1CYP1A1CYP1A2
Nonacosane SCHEMBL28207166 0.74 ABCB1 (0.83) MAOAABCB1CYP1B1CYP1A1CYP1A2
SCHEMBL9733059 0.74 ABCB1 (0.57) MAOAABCB1CYP1B1CYP1A1CYP1A2
SCHEMBL9733091 0.72 ABCB1 (0.53) MAOAABCB1CYP1B1CYP1A1CYP1A2
SCHEMBL9019328 0.72 ADORA3 (0.49) CYP3A4KDM4EMEN1MAPTKMT2A
SCHEMBL28315058 0.71 CYP3A4 (0.74) MAOAABCB1CYP1B1CYP1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0450588-B1 Substituted 3-thia- or 3-oxa-alkyl flavones, process for their preparation, their application and drugs based on these compounds as well as intermediates HOECHST AG (DE) 1996-02-28 EP disclosed
EP-0450588-A1 Substituted 3-thia- or 3-oxa-alkyl flavones, process for their preparation, their application and drugs based on these compounds as well as intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1991-10-09 EP disclosed