SCHEMBL9019366

SCHEMBL9019366

COc1ccc(-c2oc3cc(O)cc(O)c3c(=O)c2CSC/C=C(\C)CC/C=C(\C)CCC=C(C)C)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.56
CYP1A1 P04798 1/20 0.53
CYP1A2 P05177 1/20 0.53
ABCB1 P08183 1/20 0.53
MAOA P21397 1/20 0.53
CYP1B1 Q16678 1/20 0.53
FTO Q9C0B1 1/20 0.53
CYP3A4 P08684 2/20 0.52
CYP2D6 P10635 2/20 0.52
MGAM O43451 4/20 0.52
GAA P10253 4/20 0.52
SI P14410 4/20 0.52
MGAM2 Q2M2H8 4/20 0.52
PTPN1 P18031 2/20 0.52
ABCG2 Q9UNQ0 2/20 0.49
TYR P14679 1/20 0.46
BCHE P06276 1/20 0.46
ACHE P22303 1/20 0.46
KDM4E B2RXH2 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9019339 0.76 MAOA (0.60) CYP19A1CYP1A1CYP1A2ABCB1MAOA
SCHEMBL6822937 0.72 CYP19A1 (1.00) CYP19A1MGAMGAASIMGAM2
SCHEMBL6822936 0.72 CYP19A1 (1.00) CYP19A1MGAMGAASIMGAM2
Kaempferide SCHEMBL29371282 0.71 CYP1A2 (1.00) CYP19A1CYP1A1CYP1A2ABCB1MAOA
Kaempferide SCHEMBL426774 0.71 CYP1A2 (1.00) CYP19A1CYP1A1CYP1A2ABCB1MAOA
SCHEMBL29580242 0.71 CYP19A1 (0.69) CYP19A1CYP1A1CYP1A2CYP1B1MGAM
Ermanin SCHEMBL2875089 0.70 CYP3A4 (1.00) CYP1A1CYP1A2ABCB1MAOACYP1B1
SCHEMBL28037283 0.70 CYP19A1 (0.69) CYP19A1MAOAMGAMGAASI
SCHEMBL6504199 0.69 CYP1B1 (0.77) CYP19A1CYP1A1CYP1A2ABCB1MAOA
Rubraxanthone SCHEMBL8664946 0.69 MGAM (0.79) CYP19A1CYP3A4CYP2D6MGAMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0450588-B1 Substituted 3-thia- or 3-oxa-alkyl flavones, process for their preparation, their application and drugs based on these compounds as well as intermediates HOECHST AG (DE) 1996-02-28 EP disclosed
US-5173498-A For treating arteriosclerosis or hypercholesterolemia HOECHST AKTIENGESELLSCHAFT (DE) 1992-12-22 US disclosed
EP-0450588-A1 Substituted 3-thia- or 3-oxa-alkyl flavones, process for their preparation, their application and drugs based on these compounds as well as intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1991-10-09 EP disclosed