SCHEMBL902009

SCHEMBL902009

CCN(C)Cc1ccc(F)c(F)c1Br

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 6/20 0.41
RIPK1 Q13546 2/20 0.36
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
MEP1B Q16820 2/20 0.31
MEP1A Q16819 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL902072 0.72 PYCR1 (0.38) PYCR1CHRNB2CHRNA4KDM4EALDH1A1
SCHEMBL12643383 0.72 RIPK1 (0.53) PYCR1RIPK1KDM4EALDH1A1
SCHEMBL12124983 0.71 KDM4E (0.57) RIPK1KDM4EALDH1A1
SCHEMBL24136880 0.69 TYR (0.41) RIPK1CHRNB2CHRNA4
SCHEMBL6489433 0.67 GPR84 (0.35) RIPK1MEP1BMEP1A
SCHEMBL6226217 0.67 PYCR1 (0.62) PYCR1CHRNB2CHRNA4KDM4EALDH1A1
SCHEMBL19859261 0.67 PRKCE (0.34) KDM4EALDH1A1MEP1B
SCHEMBL18611210 0.66 GABRA1 (0.44) RIPK1MEP1BMEP1A
SCHEMBL23374698 0.65 RIPK1 (0.47) PYCR1RIPK1CHRNB2CHRNA4KDM4E
SCHEMBL313506 0.65 CES2 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2621919-A1 PHENYLQUINAZOLINE DERIVATIVES Merck Patent GmbH (DE) 2013-08-07 EP disclosed
WO-2012041435-A1 PHENYLQUINAZOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2012-04-05 WO disclosed