SCHEMBL9023458

SCHEMBL9023458

O=C1c2c(noc2-c2cccc(F)c2)CCC1CCCCl

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HTR1A P08908 1/20 0.32
DRD2 P14416 1/20 0.32
HTR2A P28223 1/20 0.32
ALOX5 P09917 1/20 0.32
ALOX5AP P20292 1/20 0.32
GRM5 P41594 7/20 0.32
GRIN2B Q13224 2/20 0.32
HTR7 P34969 1/20 0.32
HTR2C P28335 1/20 0.31
GRM2 Q14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9024345 0.81 HTR7 (0.43) HTR1ADRD2HTR2AGRM5HTR7
SCHEMBL9023822 0.70 HTR2A (0.39) DRD2HTR2AHTR7HTR2C
SCHEMBL9023952 0.66 HTR7 (0.41) DRD2HTR2AHTR7HTR2C
SCHEMBL9445148 0.64 HTR2A (0.40) SMN1; SMN2L3MBTL1ALDH1A1HPGDNPSR1
SCHEMBL9025048 0.63 BRD4 (0.31)
SCHEMBL9445139 0.60 HDAC1 (0.41) HTR1ADRD2HTR2AGRM5HTR7
SCHEMBL9023900 0.60 PTGS2 (0.37) ALDH1A1
SCHEMBL22449890 0.58 SMN1; SMN2 (0.40) SMN1; SMN2L3MBTL1ALDH1A1HPGDHTR1A
SCHEMBL14923166 0.56 SMN1; SMN2 (0.46) SMN1; SMN2L3MBTL1GRM5HTR7
SCHEMBL20547288 0.56 LMNA (0.50) SMN1; SMN2ALDH1A1HPGDNPSR1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0474012-B1 6,7-Dihydro-3-phenyl-1,2-benzisoxazol-4(5H)-ones and -ols, a process for their preparation and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1996-11-27 EP disclosed
US-5256672-A Antipsychotic, analgesic HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-10-26 US disclosed
US-5180834-A Antipsychotic agents HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-01-19 US disclosed
US-5114936-A Antipsychotic and analgesic agents HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-05-19 US disclosed
EP-0474012-A1 6,7-Dihydro-3-phenyl-1,2-benzisoxazol-4(5H)-ones and -ols, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-03-11 EP disclosed