SCHEMBL9023952

SCHEMBL9023952

O=C1c2c(-c3ccccc3F)noc2CCC1CCCCl

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.41
PTGS1 P23219 1/20 0.34
CYP19A1 P11511 2/20 0.32
RORC P51449 2/20 0.32
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
GABRA5 P31644 1/20 0.31
GPBAR1 Q8TDU6 1/20 0.30
DRD2 P14416 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9024867 0.93 HTR7 (0.43) HTR7PTGS1CYP19A1RORCNPC1
SCHEMBL9024797 0.84 HTR7 (0.36) HTR7PTGS1CYP19A1DRD2HTR2A
SCHEMBL9023822 0.82 HTR2A (0.39) HTR7GABRA5DRD2HTR2AHTR2C
SCHEMBL9687914 0.81 HTR7 (0.42) HTR7PTGS1RORCNPC1RAB9A
SCHEMBL9024561 0.81 HTR1A (0.45) HTR7DRD2HTR2AHTR2C
SCHEMBL9024345 0.81 HTR7 (0.43) HTR7GABRA5GPBAR1DRD2HTR2A
Hydrochloric Acid SCHEMBL9024965 0.80 HTR7 (0.41) HTR7PTGS1RORCNPC1RAB9A
SCHEMBL9024223 0.80 HTR2C (0.50) HTR7DRD2HTR2AHTR2C
SCHEMBL9024282 0.79 HTR7 (0.42) HTR7DRD2HTR2AHTR2C
SCHEMBL9445148 0.79 HTR2A (0.40) HTR7GABRA5HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0474012-B1 6,7-Dihydro-3-phenyl-1,2-benzisoxazol-4(5H)-ones and -ols, a process for their preparation and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1996-11-27 EP disclosed
US-5256672-A Antipsychotic, analgesic HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-10-26 US disclosed
US-5180834-A Antipsychotic agents HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-01-19 US disclosed
US-5114936-A Antipsychotic and analgesic agents HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-05-19 US disclosed
EP-0474012-A1 6,7-Dihydro-3-phenyl-1,2-benzisoxazol-4(5H)-ones and -ols, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-03-11 EP disclosed