SCHEMBL9023716

SCHEMBL9023716

O=C(OC1(c2ccccn2)CCNCC1)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.38
ALDH1A1 P00352 3/20 0.38
HSD17B10 Q99714 3/20 0.38
CYP3A4 P08684 3/20 0.38
CYP2D6 P10635 3/20 0.38
HPGD P15428 2/20 0.38
USP2 O75604 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MEN1 O00255 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP1A2 P05177 2/20 0.36
HSD11B1 P28845 2/20 0.35
ADORA2A P29274 1/20 0.33
TACR1 P25103 1/20 0.33
SYK P43405 1/20 0.32
POLB P06746 1/20 0.32
OPRM1 P35372 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL9023712 0.76 OPRM1 (0.49) TSHRALDH1A1HSD17B10CYP3A4CYP2D6
SCHEMBL3905108 0.75 HSD17B10 (0.41) TSHRALDH1A1HSD17B10CYP3A4CYP2D6
SCHEMBL27666393 0.72 ADRB1 (0.40) ALDH1A1MAPK1TACR1SYK
SCHEMBL7426632 0.70 HSD11B1 (0.43) TSHRALDH1A1HSD17B10CYP3A4CYP2D6
SCHEMBL21479939 0.69 ALDH1A1 (0.40) TSHRALDH1A1HSD17B10CYP3A4HPGD
Hydrochloric Acid SCHEMBL8353054 0.69 HSD11B1 (0.42) TSHRALDH1A1HSD17B10CYP3A4CYP2D6
SCHEMBL8636435 0.69 OPRM1 (0.44) TSHRALDH1A1HSD17B10CYP3A4CYP2D6
SCHEMBL29602661 0.69 OPRM1 (0.53) TSHRALDH1A1HSD17B10CYP3A4CYP2D6
SCHEMBL2222591 0.69 ALDH1A1 (0.46) TSHRALDH1A1HSD17B10CYP3A4CYP2D6
SCHEMBL171507 0.69 OPRM1 (0.53) TSHRALDH1A1HSD17B10CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0463810-B1 Heterocyclic compound and psychopharmaceutical composition containing same SUNTORY LTD (JP) 1996-01-10 EP disclosed
US-5158947-A CONDENSED HETEROCYCLIC COMPOUNDS AND PSYCHOPHARMACEUTICAL COMPOSITION CONTAINING SAME SUNTORY LIMITED (JP) 1992-10-27 US disclosed
EP-0463810-A1 Heterocyclic compound and psychopharmaceutical composition containing same SUNTORY LIMITED (JP) 1992-01-02 EP disclosed