SCHEMBL9024845

SCHEMBL9024845

O=C1COc2ccccc2C(=O)N1CCCCN1CCC(c2ccccn2)CC1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 7/20 0.48
DRD2 P14416 4/20 0.48
KCNH2 Q12809 3/20 0.48
HTR2A P28223 2/20 0.46
MCHR1 Q99705 2/20 0.46
HTR1A P08908 1/20 0.46
CHRM2 P08172 1/20 0.44
CHRM4 P08173 1/20 0.44
CHRM5 P08912 1/20 0.44
CHRM3 P20309 1/20 0.44
ADRA1A P35348 1/20 0.44
HRH1 P35367 1/20 0.44
ADRA1B P35368 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9023702 0.84 HTR7 (0.57) CHRM1DRD2KCNH2HTR2AMCHR1
SCHEMBL9024252 0.83 HTR7 (0.56) CHRM1DRD2KCNH2HTR2AMCHR1
SCHEMBL6169077 0.82 HTR1A (0.44) DRD2HTR2AHTR1AADRA1AADRA1B
SCHEMBL9371795 0.82 DRD2 (0.64) DRD2KCNH2HTR2AHTR1A
SCHEMBL31013504 0.81 HTR1A (0.71) DRD2HTR2AHTR1AADRA1AADRA1B
SCHEMBL9370364 0.81 HTR1A (0.71) DRD2HTR2AHTR1AADRA1AADRA1B
SCHEMBL9029235 0.81 ADRB2 (0.49) CHRM1DRD2CHRM2CHRM4CHRM5
SCHEMBL9372589 0.81 HTR1A (0.69) DRD2HTR2AHTR1AADRA1AADRA1B
SCHEMBL9372762 0.81 DRD3 (0.61) DRD2HTR2AHTR1AADRA1AADRA1B
SCHEMBL7472750 0.80 DRD4 (0.42) DRD2HTR1AADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0463810-B1 Heterocyclic compound and psychopharmaceutical composition containing same SUNTORY LTD (JP) 1996-01-10 EP disclosed
US-5158947-A CONDENSED HETEROCYCLIC COMPOUNDS AND PSYCHOPHARMACEUTICAL COMPOSITION CONTAINING SAME SUNTORY LIMITED (JP) 1992-10-27 US disclosed
EP-0463810-A1 Heterocyclic compound and psychopharmaceutical composition containing same SUNTORY LIMITED (JP) 1992-01-02 EP disclosed