SCHEMBL9024849

SCHEMBL9024849

Cc1noc2c1C(=O)CCC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.42
ALDH1A1 P00352 3/20 0.42
TSHR P16473 2/20 0.39
BRD4 O60885 2/20 0.38
HTT P42858 2/20 0.36
CYP1A2 P05177 2/20 0.35
CYP2C9 P11712 1/20 0.35
HTR2A P28223 4/20 0.34
HTR1A P08908 3/20 0.34
DRD2 P14416 3/20 0.34
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32
PTK2 Q05397 1/20 0.32
HPGD P15428 2/20 0.31
HSD17B10 Q99714 1/20 0.31
OPRM1 P35372 1/20 0.31
MAPT P10636 2/20 0.31
KMT2A Q03164 1/20 0.31
NPC1 O15118 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3131565 0.96 SMN1; SMN2 (0.42) SMN1; SMN2ALDH1A1TSHRBRD4HTT
SCHEMBL13145564 0.88 BRD4 (0.41) SMN1; SMN2BRD4HTR2AHTR1ADRD2
SCHEMBL21614780 0.76 BRD4 (0.41) BRD4CYP1A2CYP2C9
SCHEMBL23080469 0.72 SMN1; SMN2 (0.47) SMN1; SMN2ALDH1A1TSHRHTTCYP1A2
SCHEMBL5725151 0.72 SMN1; SMN2 (0.53) SMN1; SMN2ALDH1A1BRD4CYP1A2CYP2C9
SCHEMBL21987985 0.69 BRD4 (0.54) BRD4HTR2AHTR1ADRD2
SCHEMBL1582995 0.68 HTR7 (0.46) SMN1; SMN2ALDH1A1BRD4HPGDHSD17B10
SCHEMBL8866040 0.68 ALDH1A1 (0.34) SMN1; SMN2ALDH1A1TSHRBRD4NR3C1
SCHEMBL3139058 0.67 SMN1; SMN2 (0.32) SMN1; SMN2ALDH1A1TSHRBRD4HTR2A
SCHEMBL9445146 0.66 HTR2A (0.50) SMN1; SMN2ALDH1A1BRD4HTR2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0474012-B1 6,7-Dihydro-3-phenyl-1,2-benzisoxazol-4(5H)-ones and -ols, a process for their preparation and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1996-11-27 EP disclosed
US-5256672-A Antipsychotic, analgesic HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-10-26 US disclosed
US-5180834-A Antipsychotic agents HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-01-19 US disclosed
US-5114936-A Antipsychotic and analgesic agents HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-05-19 US disclosed
EP-0474012-A1 6,7-Dihydro-3-phenyl-1,2-benzisoxazol-4(5H)-ones and -ols, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-03-11 EP disclosed